Target Details
| UniProt AC | P42681 |
|---|---|
| Gene Symbol | TXK |
| Protein Name | Tyrosine-protein kinase TXK |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07714 (PK_Tyr_Ser-Thr) PF00017 (SH2) PF00018 (SH3_1) |
Summary
- Multi-target molecules 419
- Clinical molecules 8
- Avg pChEMBL 7.88
KEGG Pathways (1)
Active Molecules (419)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
LCFFREMLXLZNHE
|
8.9 | IC50 | 5 | — | |
MLHBMGYXWLXXSQ
|
8.9 | IC50 | 2 | — | |
NNGVMERLTTVLQP
|
8.9 | IC50 | 8 | — | |
YVYRAZLGYSUUTD
|
8.9 | IC50 | 2 | — | |
HMVGVAPFAUSEKV
|
8.9 | IC50 | 2 | — | |
KJQXTLMOVWJDQS
|
8.9 | IC50 | 4 | — | |
LAPLTIZCBMPGSJ
|
8.9 | IC50 | 2 | — | |
LFUKUCJDMFHUGZ
|
8.9 | IC50 | 3 | — | |
SOJIEOAQJTWQFG
|
8.9 | IC50 | 4 | — | |
SMOPKEHQPPXRSH
|
8.8 | IC50 | 8 | — | |
BUNVZNMOFRWGMI
|
8.8 | IC50 | 6 | — | |
QDMFSFAITDIPAB
|
8.8 | IC50 | 4 | — | |
RUJXZEMAANBOCH
|
8.8 | IC50 | 2 | — | |
BQFHXEUTDPRCLM
|
8.8 | IC50 | 4 | — | |
ZUCOXLCXLDBNCN
|
8.8 | IC50 | 4 | — | |
BFEZWHKJXGSMTK
|
8.8 | IC50 | 4 | — | |
VKQPGLDQSGLMMO
|
8.8 | IC50 | 4 | — | |
PAGIYVTUUQGTOU
|
8.7 | IC50 | 4 | — | |
PWISMKGZBHMEFG
|
8.7 | IC50 | 6 | — | |
BTWVWABAWDKQNJ
|
8.7 | IC50 | 8 | — | |
FCMIFOFGOGNZLW
|
8.7 | IC50 | 4 | — | |
BRQGUSSZIKXSNM
|
8.7 | IC50 | 3 | — | |
LHFAKDSSXLAPAE
|
8.7 | IC50 | 4 | — | |
RVKCUGLKWDUXGI
|
8.7 | IC50 | 4 | — | |
COPLBPVGYVVHTD
|
8.7 | IC50 | 2 | — | |
NGZPCPROZUYFJJ
|
8.7 | IC50 | 6 | — | |
VYVIHHSHQWYIAI
|
8.7 | IC50 | 3 | — | |
ZBNZXTGUTAYRHI
|
8.7 | Kd | 102 | Yes | |
AESJMHXIUSDHBC
|
8.7 | IC50 | 4 | — | |
PZWSKESWDIFAFK
|
8.7 | IC50 | 9 | — | |
GZDQSSZYDSPMRO
|
8.7 | IC50 | 3 | — | |
GOOMNGHXGYAHJM
|
8.6 | IC50 | 7 | — | |
RZSSIBVYFFJHNU
|
8.6 | IC50 | 4 | — | |
XYFPWWZEPKGCCK
|
8.6 | IC50 | 7 | — | |
DFNGRDVXGRSFSL
|
8.6 | IC50 | 3 | — | |
XYFPWWZEPKGCCK
|
8.6 | IC50 | 34 | — | |
CRYRQUNNVGZTRP
|
8.6 | IC50 | 4 | — | |
KJRVCMVPIKELBC
|
8.6 | IC50 | 12 | — | |
NCJOAUQODQCQHX
|
8.6 | IC50 | 3 | — | |
XXJWOZLYIDMCJH
|
8.6 | IC50 | 4 | — | |
ZNGBTVQWFICDEF
|
8.6 | IC50 | 4 | — | |
KUWNIYPIWGNUOY
|
8.6 | IC50 | 4 | — | |
RCDQXYOSLXRXQP
|
8.5 | IC50 | 4 | — | |
DJKOMFSZAABEBE
|
8.5 | IC50 | 4 | — | |
RNOAOAWBMHREKO
|
8.5 | IC50 | 15 | — | |
FTMHKFYFKGDOSY
|
8.5 | IC50 | 3 | — | |
SRSNLQWDLJRJNW
|
8.5 | IC50 | 4 | — | |
UDQYLBAFAGJAOD
|
8.5 | IC50 | 2 | — | |
WXXZWHIGBFHJJG
|
8.5 | IC50 | 3 | — | |
IBELJEQCPODFNE
|
8.5 | IC50 | 4 | — |