Target Details
| UniProt AC | P42681 |
|---|---|
| Gene Symbol | TXK |
| Protein Name | Tyrosine-protein kinase TXK |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07714 (PK_Tyr_Ser-Thr) PF00017 (SH2) PF00018 (SH3_1) |
Summary
- Multi-target molecules 419
- Clinical molecules 8
- Avg pChEMBL 7.88
KEGG Pathways (1)
Active Molecules (419)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
STTWMUJSAKOTEV
|
9.4 | IC50 | 4 | — | |
JKTAWSRABQDLCF
|
9.4 | IC50 | 4 | — | |
PFZFZZIBHZGYGR
|
9.4 | IC50 | 4 | — | |
ACWBHJAIEPRBBS
|
9.4 | IC50 | 4 | — | |
CWBFGXHQESGYOA
|
9.4 | IC50 | 4 | — | |
FHSFSZVDXBNGIW
|
9.3 | IC50 | 4 | — | |
NQMUJZRUULJLJA
|
9.3 | IC50 | 4 | — | |
CRYRQUNNVGZTRP
|
9.3 | IC50 | 4 | — | |
SEBXKXKMNLLVGQ
|
9.3 | IC50 | 3 | — | |
UNRUSKKHCUBUIG
|
9.3 | IC50 | 4 | — | |
WFTDUNFLISNELR
|
9.3 | IC50 | 4 | — | |
YEQGARBJDLREPV
|
9.3 | IC50 | 4 | — | |
MTQFNASJEDTODL
|
9.3 | IC50 | 4 | — | |
WQIKESWJRYQGPJ
|
9.3 | IC50 | 3 | — | |
BLPMXZJSJLHCPQ
|
9.3 | IC50 | 2 | — | |
FHRWBUZVAOTINV
|
9.3 | IC50 | 4 | — | |
KWLMYZZUWSGKCI
|
9.3 | IC50 | 4 | — | |
UQPCMSBCSBHRAK
|
9.3 | IC50 | 4 | — | |
BGHWKOZZYSOJOH
|
9.2 | IC50 | 4 | — | |
DAXOKBQPWOTXRO
|
9.2 | IC50 | 4 | — | |
IHIHUZCUZXZSPC
|
9.2 | IC50 | 4 | — | |
JWCAOJUUMHNEDQ
|
9.2 | IC50 | 4 | — | |
DEZYACNEATUTOK
|
9.2 | IC50 | 4 | — | |
BOXWOAGQDNNJAR
|
9.2 | IC50 | 4 | — | |
PWBFGGSRGAQQKP
|
9.2 | IC50 | 4 | — | |
WLIPXINLXDDYNF
|
9.2 | IC50 | 4 | — | |
UITFXMJLCNZEOF
|
9.2 | IC50 | 2 | — | |
KCRLEHJVPAGRCS
|
9.2 | IC50 | 4 | — | |
KORMETUWFBVJKV
|
9.1 | IC50 | 4 | — | |
KITSIKGMHVEYCU
|
9.1 | IC50 | 4 | — | |
NDBOXIGFGPEIBN
|
9.1 | IC50 | 4 | — | |
VMQYRLKWZIILQI
|
9.1 | IC50 | 4 | — | |
QLJUTZNCZYGNKW
|
9.1 | IC50 | 4 | — | |
ZJZHIMCDAFDFRU
|
9.1 | IC50 | 3 | — | |
ZKLWHHZNVMVOLN
|
9.1 | IC50 | 2 | — | |
LAPLTIZCBMPGSJ
|
9.1 | IC50 | 2 | — | |
RUJXZEMAANBOCH
|
9.1 | IC50 | 2 | — | |
MSIACRQJKTVOPV
|
9.0 | IC50 | 4 | — | |
DPIFGUKPQIBTRZ
|
9.0 | IC50 | 3 | — | |
QALLXGXAWLTZAF
|
9.0 | IC50 | 4 | — | |
ZMBXNTKDEKXKSP
|
9.0 | IC50 | 4 | — | |
FENGJEKSOMGGKU
|
9.0 | IC50 | 4 | — | |
OZLQMOHHARKWIF
|
9.0 | IC50 | 4 | — | |
SDBRHZQODRZNMB
|
9.0 | IC50 | 4 | — | |
YFKVYBRENKNUCS
|
9.0 | IC50 | 4 | — | |
ATYAIDXPSYJANV
|
9.0 | IC50 | 4 | — | |
KKDKMWVZUKAQOJ
|
9.0 | IC50 | 4 | — | |
DFAZTCINNFBPMC
|
9.0 | IC50 | 4 | — | |
MPLZFNKPADDSLE
|
8.9 | IC50 | 4 | — | |
NUTQNNLZHMFJOK
|
8.9 | IC50 | 4 | — |