Target Details
| UniProt AC | P42681 |
|---|---|
| Gene Symbol | TXK |
| Protein Name | Tyrosine-protein kinase TXK |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07714 (PK_Tyr_Ser-Thr) PF00017 (SH2) PF00018 (SH3_1) |
Summary
- Multi-target molecules 419
- Clinical molecules 8
- Avg pChEMBL 7.88
KEGG Pathways (1)
Active Molecules (419)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
MOKNRUDQTSPKQC
|
9.9 | IC50 | 3 | — | |
KBEOUCGXJVQSTA
|
9.8 | IC50 | 4 | — | |
SJYAVQZFEBVYGJ
|
9.8 | IC50 | 4 | — | |
CSRJXMBBNXGWNS
|
9.8 | IC50 | 4 | — | |
XGOJEPJETCHLMD
|
9.8 | IC50 | 4 | — | |
NHMAKMLWAUSTMS
|
9.7 | IC50 | 4 | — | |
QBTKIUOSXLNHIK
|
9.7 | IC50 | 4 | — | |
QPIYIWYNEVEBBY
|
9.7 | IC50 | 4 | — | |
BLPMXZJSJLHCPQ
|
9.7 | IC50 | 2 | — | |
FHNCSRKSWPZETL
|
9.7 | IC50 | 4 | — | |
MSOXGTBOMYQLRK
|
9.7 | IC50 | 4 | — | |
UBWXSCATULGCSA
|
9.7 | IC50 | 4 | — | |
WPFZWTKQXNTKQJ
|
9.7 | IC50 | 4 | — | |
ZKLWHHZNVMVOLN
|
9.7 | IC50 | 2 | — | |
AKAMMFZEIZKQBD
|
9.7 | IC50 | 4 | — | |
FINZRTUQZUBKBD
|
9.7 | IC50 | 4 | — | |
UHNKAVIIGHQZAC
|
9.7 | IC50 | 3 | — | |
CQYOCHGVYYCAJH
|
9.7 | IC50 | 4 | — | |
KNEKVQSXRQKRBO
|
9.7 | IC50 | 4 | — | |
SUHPRCQYTXOSRF
|
9.7 | IC50 | 4 | — | |
GFGUDIMDIZPFBT
|
9.6 | IC50 | 3 | — | |
YWBAOBYDVWSCMN
|
9.6 | IC50 | 4 | — | |
QRYWETQFXDSLKP
|
9.6 | IC50 | 4 | — | |
BQFHXEUTDPRCLM
|
9.6 | IC50 | 4 | — | |
DFNGRDVXGRSFSL
|
9.6 | IC50 | 2 | — | |
PUZRMPODDLWRDD
|
9.6 | IC50 | 3 | — | |
NFVGAIXPTCGYPB
|
9.6 | IC50 | 2 | — | |
BUXSSQZWDXOIAY
|
9.5 | IC50 | 4 | — | |
CYGPGKKCJOVFQJ
|
9.5 | IC50 | 4 | — | |
MOWYXIYUNCUBBO
|
9.5 | IC50 | 4 | — | |
LZOYRTMQLOFTSF
|
9.5 | IC50 | 4 | — | |
OJNRDLFIHPXKMH
|
9.5 | IC50 | 2 | — | |
OJNRDLFIHPXKMH
|
9.5 | IC50 | 2 | — | |
YZJBXGLZGKPCPE
|
9.5 | IC50 | 2 | — | |
ZEJMFFQWPNGDLL
|
9.5 | IC50 | 2 | — | |
WPKTWCDIDXHHLT
|
9.5 | IC50 | 2 | — | |
DLWDBHBTVQQBJZ
|
9.5 | IC50 | 4 | — | |
UNSFWPUQRXYWKE
|
9.5 | IC50 | 4 | — | |
ZUXIOCJCONDJBE
|
9.5 | IC50 | 4 | — | |
OXVXVYNMDOKNGH
|
9.5 | IC50 | 3 | — | |
AMWYKVLLDVPZKH
|
9.5 | IC50 | 3 | — | |
NHMAKMLWAUSTMS
|
9.5 | IC50 | 3 | — | |
OZAGVJOYZGRSJN
|
9.5 | IC50 | 4 | — | |
FMUGXGTXXNULGS
|
9.4 | IC50 | 4 | — | |
IZIBDTDSPVBIEA
|
9.4 | IC50 | 4 | — | |
ZECYSSILAXMSLF
|
9.4 | IC50 | 3 | — | |
GFXJEHXKSRGUJJ
|
9.4 | IC50 | 4 | — | |
RXBBNYOZZYEKJZ
|
9.4 | IC50 | 4 | — | |
WASKPESMKKPPGO
|
9.4 | IC50 | 4 | — | |
LKLIRPMEYRVLFV
|
9.4 | IC50 | 3 | — |