Target Details
| UniProt AC | P42680 |
|---|---|
| Gene Symbol | TEC |
| Protein Name | Tyrosine-protein kinase Tec |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00779 (BTK) PF00169 (PH) PF07714 (PK_Tyr_Ser-Thr) PF00017 (SH2) PF00018 (SH3_1) |
Summary
- Multi-target molecules 309
- Clinical molecules 7
- Avg pChEMBL 7.78
KEGG Pathways (2)
Active Molecules (309)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
VAARYSWULJUGST
|
6.2 | Kd | 119 | Yes | |
SFMJNHNUOVADRW
|
6.2 | IC50 | 7 | — | |
LCVIRAZGMYMNNT
|
6.2 | Kd | 20 | — | |
HHFBDROWDBDFBR
|
6.1 | Kd | 40 | Yes | |
FLBNLJLONKAPLR
|
6.0 | Kd | 31 | — | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — | |
KDKUVYLMPJIGKA
|
6.0 | Kd | 91 | Yes | |
KHVVJKLNKLQLJZ
|
6.0 | IC50 | 288 | — | |
MAHFVAHPQSLLJF
|
6.0 | IC50 | 288 | — |