Target Details
| UniProt AC | P42680 |
|---|---|
| Gene Symbol | TEC |
| Protein Name | Tyrosine-protein kinase Tec |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00779 (BTK) PF00169 (PH) PF07714 (PK_Tyr_Ser-Thr) PF00017 (SH2) PF00018 (SH3_1) |
Summary
- Multi-target molecules 309
- Clinical molecules 7
- Avg pChEMBL 7.78
KEGG Pathways (2)
Active Molecules (309)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
AHBFBRPGNOVEBK
|
6.8 | IC50 | 11 | — | |
CZSSHLOWZFKWML
|
6.8 | IC50 | 3 | — | |
LSJWYMSFUWBGPN
|
6.8 | IC50 | 17 | — | |
PWDHQTXOIXSDBN
|
6.8 | IC50 | 2 | — | |
NVDXHXCRQAOJQR
|
6.8 | IC50 | 2 | — | |
KPZGJWPPVXZLDN
|
6.7 | IC50 | 10 | — | |
QQWUGDVOUVUTOY
|
6.7 | Kd | 231 | Yes | |
GZYUJXFTHLKPAK
|
6.7 | IC50 | 16 | — | |
LXOADFXFUMUSSE
|
6.7 | IC50 | 3 | — | |
RTRNJQOBEOISFQ
|
6.7 | IC50 | 5 | — | |
WNEODWDFDXWOLU
|
6.7 | Kd | 5 | — | |
ZFDGMDVYMNWICG
|
6.7 | IC50 | 2 | — | |
GEEUDEOZMWBPDT
|
6.7 | IC50 | 4 | — | |
OPKHZFMFWCMAPS
|
6.7 | IC50 | 6 | — | |
MZSDTUIZKGUVHK
|
6.6 | IC50 | 4 | — | |
RFCJOYPMBVRHBV
|
6.6 | IC50 | 5 | — | |
LAUHLGUSVSJYCI
|
6.6 | IC50 | 16 | — | |
HGYLDYXQKAISMX
|
6.6 | Kd | 4 | — | |
JSAQBOQCZJHWMA
|
6.6 | Kd | 11 | — | |
RRDIEPDENZRYJK
|
6.6 | IC50 | 3 | — | |
DPRNXTSMYVCYLJ
|
6.6 | IC50 | 13 | — | |
WMMNTQFZCHUZSM
|
6.6 | IC50 | 14 | — | |
UBPYILGKFZZVDX
|
6.5 | IC50 | 130 | Yes | |
WKDACQVEJIVHMZ
|
6.5 | Kd | 46 | — | |
HUFOZJXAKZVRNJ
|
6.5 | Kd | 10 | — | |
SXKQCOANBPFCHG
|
6.5 | IC50 | 3 | — | |
FHOKFOHRQUSPMF
|
6.5 | IC50 | 3 | — | |
CXQHYVUVSFXTMY
|
6.5 | Kd | 154 | — | |
SEJGTFPOEJWEGG
|
6.5 | Kd | 149 | — | |
YFVRNHCFDWIILZ
|
6.5 | IC50 | 3 | — | |
DUYJMQONPNNFPI
|
6.5 | Kd | 11 | — | |
XZAATUBTUPPERZ
|
6.5 | IC50 | 6 | — | |
SRXKFAPDNBKKAP
|
6.5 | IC50 | 2 | — | |
VTJHGMZHVOXJPG
|
6.4 | IC50 | 15 | — | |
VXJXHNMYRAHBBO
|
6.4 | IC50 | 5 | — | |
ZAJXXUDARPGGOC
|
6.4 | Kd | 4 | — | |
ZJSNZHATZAWKIQ
|
6.4 | Kd | 5 | — | |
UAXCBCHLHXDOSO
|
6.4 | IC50 | 2 | — | |
WDTHDWKPTWWHLS
|
6.4 | IC50 | 13 | — | |
BCPNJXKITYKKCV
|
6.3 | IC50 | 2 | — | |
CFYBPLINLQYRJH
|
6.3 | IC50 | 2 | — | |
CZXXHLKIPJUICC
|
6.3 | IC50 | 2 | — | |
KEVGNTLGNXQCTI
|
6.3 | IC50 | 2 | — | |
KKOFOOADVSUXAK
|
6.3 | IC50 | 3 | — | |
LAVICBXNQHDFND
|
6.3 | IC50 | 3 | — | |
LJKHVTUWGNPBJV
|
6.3 | IC50 | 3 | — | |
PGVGTJDOYNQGLQ
|
6.3 | IC50 | 2 | — | |
UULCMWFOJYIYAC
|
6.3 | IC50 | 3 | — | |
YOVVNQKCSKSHKT
|
6.2 | Kd | 15 | — | |
CBRJPFGIXUFMTM
|
6.2 | IC50 | 7 | — |