Target Details
| UniProt AC | P42680 |
|---|---|
| Gene Symbol | TEC |
| Protein Name | Tyrosine-protein kinase Tec |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00779 (BTK) PF00169 (PH) PF07714 (PK_Tyr_Ser-Thr) PF00017 (SH2) PF00018 (SH3_1) |
Summary
- Multi-target molecules 309
- Clinical molecules 7
- Avg pChEMBL 7.78
KEGG Pathways (2)
Active Molecules (309)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ILXFYIOJPFUYGX
|
7.2 | IC50 | 5 | — | |
IRMJEKARXQRXOY
|
7.2 | IC50 | 3 | — | |
PTHVKCSYXICMAR
|
7.2 | IC50 | 14 | — | |
HEFUQOMXBZIABJ
|
7.2 | IC50 | 2 | — | |
IZQVCAWYZWMWJS
|
7.2 | IC50 | 4 | — | |
GOLVRUHMODBSGJ
|
7.2 | IC50 | 3 | — | |
JUSWPUDQOKINJO
|
7.2 | IC50 | 16 | — | |
OPHSZSZDICRBPP
|
7.2 | IC50 | 16 | — | |
SRSQULBCTWSVKL
|
7.2 | IC50 | 15 | — | |
FTWCGCABDYPPKS
|
7.2 | IC50 | 4 | — | |
ZZJOFPXLPFXEKV
|
7.2 | IC50 | 4 | — | |
QRIXKWMQRHCONV
|
7.2 | IC50 | 4 | — | |
DOVHWPFJHQGYDS
|
7.2 | IC50 | 4 | — | |
OMIQRSKHABIPRH
|
7.2 | IC50 | 15 | — | |
DKCAHMDAWGVHSL
|
7.2 | Kd | 3 | — | |
LPFWVDIFUFFKJU
|
7.2 | Kd | 9 | — | |
XYFZVVYVIFJBIS
|
7.2 | IC50 | 17 | — | |
NMNLVTJEQAQJHN
|
7.1 | IC50 | 4 | — | |
MCDRCFIVCSZLRU
|
7.1 | IC50 | 3 | — | |
TUMDRAALZUBTGH
|
7.1 | IC50 | 3 | — | |
IHJOVKPLSQINCA
|
7.1 | IC50 | 3 | — | |
LCYSSHSIKSARGO
|
7.1 | IC50 | 19 | — | |
XYFPWWZEPKGCCK
|
7.1 | IC50 | 7 | — | |
NVDXHXCRQAOJQR
|
7.1 | IC50 | 3 | — | |
ZYQIUDPJBOUHCC
|
7.1 | IC50 | 4 | — | |
ATLOUNJJIAISOI
|
7.0 | IC50 | 4 | — | |
CDISOBGWDHAHGF
|
7.0 | IC50 | 16 | — | |
UBUVIQYWARUKMQ
|
7.0 | IC50 | 4 | — | |
WDENQIQQYWYTPO
|
7.0 | IC50 | 8 | — | |
SRXKFAPDNBKKAP
|
7.0 | IC50 | 2 | — | |
LUMAVJBHSUJPOG
|
7.0 | IC50 | 4 | — | |
ZFDGMDVYMNWICG
|
7.0 | IC50 | 10 | — | |
SSDFTYWIYVWCIE
|
7.0 | IC50 | 17 | — | |
ZMCYWNHBOFVQPF
|
7.0 | IC50 | 3 | — | |
BBDSYVIXESVDPE
|
7.0 | IC50 | 4 | — | |
CUABMPOJOBCXJI
|
7.0 | Kd | 3 | — | |
OSAWFUCUZJNEID
|
6.9 | IC50 | 20 | — | |
SDVAHCXGDGYWFA
|
6.9 | IC50 | 12 | — | |
KRILZVCKKUOPKH
|
6.9 | IC50 | 4 | — | |
WZLCFQWCRHXUJG
|
6.9 | IC50 | 4 | — | |
CVBABGVEYUMHNU
|
6.9 | IC50 | 6 | — | |
BLOSAGLLXHJECN
|
6.9 | IC50 | 4 | — | |
GKZGJDDKZTVQJZ
|
6.9 | IC50 | 4 | — | |
UBXMXLKDIBLSPB
|
6.9 | IC50 | 3 | — | |
LBCWQLSBINGIBS
|
6.9 | IC50 | 2 | — | |
LOLPPWBBNUVNQZ
|
6.9 | Kd | 97 | Yes | |
XQMGYYWEPWXCJB
|
6.8 | IC50 | 2 | — | |
NFLKTKKJFVNGLH
|
6.8 | IC50 | 4 | — | |
VQUUBQYYHFHNFA
|
6.8 | IC50 | 4 | — | |
UMBDWDIRLTVPBF
|
6.8 | IC50 | 9 | — |