Target Details
| UniProt AC | P42680 |
|---|---|
| Gene Symbol | TEC |
| Protein Name | Tyrosine-protein kinase Tec |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00779 (BTK) PF00169 (PH) PF07714 (PK_Tyr_Ser-Thr) PF00017 (SH2) PF00018 (SH3_1) |
Summary
- Multi-target molecules 309
- Clinical molecules 7
- Avg pChEMBL 7.78
KEGG Pathways (2)
Active Molecules (309)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
OZLQMOHHARKWIF
|
7.8 | IC50 | 4 | — | |
KCRLEHJVPAGRCS
|
7.8 | IC50 | 4 | — | |
WIZIQUFUGUEWKY
|
7.8 | IC50 | 6 | — | |
RNOAOAWBMHREKO
|
7.8 | IC50 | 15 | — | |
BFEZWHKJXGSMTK
|
7.7 | IC50 | 4 | — | |
MNDLPZPZVIEBFF
|
7.7 | IC50 | 4 | — | |
ZTUJNJAKTLHBEX
|
7.7 | IC50 | 5 | — | |
QNNJMWIVIVLSHC
|
7.7 | IC50 | 4 | — | |
QUIWHXQETADMGN
|
7.7 | IC50 | 4 | — | |
VSFINVOSLLRTIP
|
7.7 | IC50 | 6 | — | |
SXLIACXIXLLKGR
|
7.7 | IC50 | 4 | — | |
DNFWTELNLRENAM
|
7.7 | IC50 | 4 | — | |
PAGIYVTUUQGTOU
|
7.7 | IC50 | 4 | — | |
ZDWLIFUKOJCBAL
|
7.7 | IC50 | 3 | — | |
NCEZXFYYHDEYFJ
|
7.6 | IC50 | 3 | — | |
FUZSHLVNKZZEKR
|
7.6 | IC50 | 16 | — | |
GXANJKDFGYJBEM
|
7.6 | IC50 | 5 | — | |
RCDQXYOSLXRXQP
|
7.5 | IC50 | 4 | — | |
OETOLISJTPMUFM
|
7.5 | Kd | 4 | — | |
ABSANYKJICYHQP
|
7.5 | IC50 | 4 | — | |
KQISOZQPFQHIFH
|
7.5 | IC50 | 4 | — | |
WCCLANJGOUJNNL
|
7.5 | IC50 | 4 | — | |
HKSZLNNOFSGOKW
|
7.5 | IC50 | 408 | — | |
MTQFNASJEDTODL
|
7.5 | IC50 | 4 | — | |
RJARQSDFMBQVEH
|
7.4 | IC50 | 4 | — | |
MZPVEMOYADUARK
|
7.4 | IC50 | 2 | — | |
HDVYJNSAOAUAIQ
|
7.4 | IC50 | 4 | — | |
VYZQSAKXLMEDCB
|
7.4 | IC50 | 9 | — | |
KOQJXUXLQGQJDF
|
7.4 | IC50 | 4 | — | |
XSNVEELQPXGAPX
|
7.4 | Kd | 3 | — | |
UQPCMSBCSBHRAK
|
7.4 | IC50 | 3 | — | |
YPXWUKLQAUBCPF
|
7.4 | IC50 | 8 | — | |
AEBADKNVNADXNA
|
7.4 | IC50 | 3 | — | |
LXURGGKEOPHREO
|
7.4 | IC50 | 13 | — | |
PZWSKESWDIFAFK
|
7.4 | IC50 | 9 | — | |
RZSSIBVYFFJHNU
|
7.4 | IC50 | 4 | — | |
WRMWTYPCAZJKRH
|
7.4 | IC50 | 3 | — | |
ALKJNCZNEOTEMP
|
7.3 | Kd | 55 | — | |
CLKNHJDZJCCLAZ
|
7.3 | IC50 | 4 | — | |
ZXGCNNKDPNECIS
|
7.3 | IC50 | 4 | — | |
DNDCQFCAXLONFM
|
7.3 | IC50 | 4 | — | |
CRYRQUNNVGZTRP
|
7.3 | IC50 | 4 | — | |
YYRYNQBAVOOSOA
|
7.3 | IC50 | 4 | — | |
GAWQIOVCXHLEAP
|
7.3 | Kd | 4 | — | |
IVUHUFVVODTZOQ
|
7.3 | Kd | 3 | — | |
VZOSDPVVDDOWFT
|
7.3 | IC50 | 2 | — | |
WDZZTNVBOLILQA
|
7.3 | IC50 | 2 | — | |
BPMZEUVOCIAUDQ
|
7.3 | IC50 | 4 | — | |
OYFVJVWLUDKTIF
|
7.3 | IC50 | 4 | — | |
TXIUPNHPXDVAAM
|
7.2 | IC50 | 5 | — |