Target Details
| UniProt AC | P42680 |
|---|---|
| Gene Symbol | TEC |
| Protein Name | Tyrosine-protein kinase Tec |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00779 (BTK) PF00169 (PH) PF07714 (PK_Tyr_Ser-Thr) PF00017 (SH2) PF00018 (SH3_1) |
Summary
- Multi-target molecules 309
- Clinical molecules 7
- Avg pChEMBL 7.78
KEGG Pathways (2)
Active Molecules (309)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
CDUYTHAOJIKLFN
|
8.3 | IC50 | 4 | — | |
SXXABOHFQFARBT
|
8.3 | IC50 | 5 | — | |
FCMIFOFGOGNZLW
|
8.3 | IC50 | 4 | — | |
FINZRTUQZUBKBD
|
8.3 | IC50 | 3 | — | |
MODKQWIWLUEOCI
|
8.3 | IC50 | 3 | — | |
ATTKNMWCPOFQHD
|
8.3 | IC50 | 2 | — | |
BYZCNAKZYXERPN
|
8.3 | IC50 | 2 | — | |
SRSNLQWDLJRJNW
|
8.3 | IC50 | 4 | — | |
KWLMYZZUWSGKCI
|
8.3 | IC50 | 4 | — | |
BOXWOAGQDNNJAR
|
8.2 | IC50 | 4 | — | |
UGBDLAMFDOZLBT
|
8.2 | IC50 | 3 | — | |
DAXOKBQPWOTXRO
|
8.2 | IC50 | 4 | — | |
KSUDUUBCXJUFRL
|
8.2 | Kd | 12 | — | |
UNRUSKKHCUBUIG
|
8.2 | IC50 | 4 | — | |
WLIPXINLXDDYNF
|
8.2 | IC50 | 4 | — | |
AHGUJKCTSXOYES
|
8.2 | IC50 | 4 | — | |
KXBDTLQSDKGAEB
|
8.2 | IC50 | 8 | — | |
SMOPKEHQPPXRSH
|
8.2 | IC50 | 8 | — | |
GFZZUAFZBKEOHV
|
8.2 | IC50 | 7 | — | |
NAXFVNQSUIOSIC
|
8.2 | IC50 | 4 | — | |
UVUTZINLTAEGAD
|
8.2 | IC50 | 4 | — | |
XYFPWWZEPKGCCK
|
8.2 | IC50 | 34 | — | |
CDFHNEWIEMNZKE
|
8.1 | IC50 | 4 | — | |
IBELJEQCPODFNE
|
8.1 | IC50 | 4 | — | |
NUDBRCUXDGGUOA
|
8.1 | IC50 | 4 | — | |
KAFKHBRCDYVZDT
|
8.1 | IC50 | 4 | — | |
KOEUOFPEZFUWRF
|
8.1 | IC50 | 4 | — | |
ZNGBTVQWFICDEF
|
8.1 | IC50 | 4 | — | |
ZMBXNTKDEKXKSP
|
8.1 | IC50 | 4 | — | |
BTWVWABAWDKQNJ
|
8.1 | IC50 | 8 | — | |
CKXVUTSXVABAMG
|
8.1 | IC50 | 4 | — | |
LHLGYQRKVKDWSY
|
8.1 | IC50 | 4 | — | |
IHIHUZCUZXZSPC
|
8.0 | IC50 | 4 | — | |
ZRYMMWAJAFUANM
|
8.0 | IC50 | 7 | — | |
AESJMHXIUSDHBC
|
8.0 | IC50 | 4 | — | |
FHSFSZVDXBNGIW
|
8.0 | IC50 | 4 | — | |
KJQXTLMOVWJDQS
|
8.0 | IC50 | 4 | — | |
SDBRHZQODRZNMB
|
8.0 | IC50 | 4 | — | |
VWYWHQKPHALPKU
|
8.0 | IC50 | 3 | — | |
MWKSRKSEWLRPBL
|
7.9 | Kd | 1075 | — | |
XYFPWWZEPKGCCK
|
7.9 | IC50 | 7 | — | |
ZCCPLJOKGAACRT
|
7.9 | Kd | 599 | — | |
OVBRVYHGBQUXHR
|
7.9 | Kd | 4 | — | |
TVJRDCQUZMGBAB
|
7.9 | IC50 | 13 | — | |
ZBNZXTGUTAYRHI
|
7.9 | Kd | 102 | Yes | |
ZEIZIRVZVXALHM
|
7.9 | IC50 | 3 | — | |
MRNPOLZRBHNDGI
|
7.9 | IC50 | 4 | — | |
IGXJXMLDIIGDNE
|
7.8 | IC50 | 8 | — | |
OXOMWFOJARKFIY
|
7.8 | IC50 | 4 | — | |
SEJLPXCPMNSRAM
|
7.8 | IC50 | 7 | — |