Target Details
| UniProt AC | P42680 |
|---|---|
| Gene Symbol | TEC |
| Protein Name | Tyrosine-protein kinase Tec |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00779 (BTK) PF00169 (PH) PF07714 (PK_Tyr_Ser-Thr) PF00017 (SH2) PF00018 (SH3_1) |
Summary
- Multi-target molecules 309
- Clinical molecules 7
- Avg pChEMBL 7.78
KEGG Pathways (2)
Active Molecules (309)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
RVKCUGLKWDUXGI
|
8.8 | IC50 | 4 | — | |
XXJWOZLYIDMCJH
|
8.8 | IC50 | 4 | — | |
NHMAKMLWAUSTMS
|
8.8 | IC50 | 4 | — | |
ZUXIOCJCONDJBE
|
8.8 | IC50 | 4 | — | |
QDMFSFAITDIPAB
|
8.8 | IC50 | 4 | — | |
VWJGTQUINXNBOY
|
8.8 | IC50 | 4 | — | |
ZUCOXLCXLDBNCN
|
8.8 | IC50 | 4 | — | |
UQPCMSBCSBHRAK
|
8.8 | IC50 | 4 | — | |
BUNVZNMOFRWGMI
|
8.7 | IC50 | 6 | — | |
KZMQPYCXSAGLTB
|
8.7 | IC50 | 8 | — | |
VKQPGLDQSGLMMO
|
8.7 | IC50 | 4 | — | |
PFZFZZIBHZGYGR
|
8.7 | IC50 | 4 | — | |
DFAZTCINNFBPMC
|
8.7 | IC50 | 4 | — | |
NGZPCPROZUYFJJ
|
8.7 | IC50 | 6 | — | |
UNSFWPUQRXYWKE
|
8.7 | IC50 | 4 | — | |
CRYRQUNNVGZTRP
|
8.7 | IC50 | 4 | — | |
LHFAKDSSXLAPAE
|
8.7 | IC50 | 4 | — | |
PWBFGGSRGAQQKP
|
8.6 | IC50 | 4 | — | |
QCJFYACTZIVZBB
|
8.6 | IC50 | 8 | — | |
FENGJEKSOMGGKU
|
8.6 | IC50 | 4 | — | |
QALLXGXAWLTZAF
|
8.6 | IC50 | 4 | — | |
BQFHXEUTDPRCLM
|
8.6 | IC50 | 4 | — | |
DJKOMFSZAABEBE
|
8.6 | IC50 | 4 | — | |
PWISMKGZBHMEFG
|
8.6 | IC50 | 6 | — | |
DLWDBHBTVQQBJZ
|
8.6 | IC50 | 4 | — | |
MSIACRQJKTVOPV
|
8.6 | IC50 | 4 | — | |
DFUIAUMNSYRTOL
|
8.5 | IC50 | 3 | — | |
IRBVGTPPFBYDKX
|
8.5 | IC50 | 9 | — | |
DQFOPMWZUFUHDC
|
8.5 | IC50 | 6 | — | |
BGHWKOZZYSOJOH
|
8.5 | IC50 | 4 | — | |
WASKPESMKKPPGO
|
8.5 | IC50 | 4 | — | |
NHMAKMLWAUSTMS
|
8.5 | IC50 | 3 | — | |
AOKKWYGSIRAXIZ
|
8.5 | IC50 | 4 | — | |
BIRLBQULISTSMZ
|
8.5 | IC50 | 4 | — | |
NUTQNNLZHMFJOK
|
8.5 | IC50 | 4 | — | |
HJAUUHMYFPHMCT
|
8.4 | IC50 | 4 | — | |
BIRLBQULISTSMZ
|
8.4 | IC50 | 3 | — | |
FMRJPPUXBYSJRE
|
8.4 | IC50 | 4 | — | |
XIDJFSRGLOUDGG
|
8.4 | IC50 | 4 | — | |
SBRIQINKAOKMMM
|
8.4 | IC50 | 6 | — | |
KUWNIYPIWGNUOY
|
8.4 | IC50 | 4 | — | |
SOJIEOAQJTWQFG
|
8.4 | IC50 | 4 | — | |
RNOAOAWBMHREKO
|
8.4 | IC50 | 3 | — | |
JWCAOJUUMHNEDQ
|
8.4 | IC50 | 4 | — | |
WFTDUNFLISNELR
|
8.4 | IC50 | 4 | — | |
KORMETUWFBVJKV
|
8.4 | IC50 | 4 | — | |
NDBOXIGFGPEIBN
|
8.3 | IC50 | 4 | — | |
NZIQNLGMMJGSQU
|
8.3 | IC50 | 6 | — | |
XNPHXLCYBBQUQK
|
8.3 | IC50 | 4 | — | |
SUHPRCQYTXOSRF
|
8.3 | IC50 | 4 | — |