Target Details
| UniProt AC | P42680 |
|---|---|
| Gene Symbol | TEC |
| Protein Name | Tyrosine-protein kinase Tec |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00779 (BTK) PF00169 (PH) PF07714 (PK_Tyr_Ser-Thr) PF00017 (SH2) PF00018 (SH3_1) |
Summary
- Multi-target molecules 309
- Clinical molecules 7
- Avg pChEMBL 7.78
KEGG Pathways (2)
Active Molecules (309)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
CSRJXMBBNXGWNS
|
10.1 | IC50 | 4 | — | |
KBEOUCGXJVQSTA
|
10.1 | IC50 | 4 | — | |
XGOJEPJETCHLMD
|
10.0 | IC50 | 4 | — | |
SJYAVQZFEBVYGJ
|
10.0 | IC50 | 4 | — | |
AKAMMFZEIZKQBD
|
9.9 | IC50 | 4 | — | |
OZAGVJOYZGRSJN
|
9.8 | IC50 | 4 | — | |
CQYOCHGVYYCAJH
|
9.8 | IC50 | 4 | — | |
QPIYIWYNEVEBBY
|
9.8 | IC50 | 4 | — | |
FHNCSRKSWPZETL
|
9.7 | IC50 | 4 | — | |
QBTKIUOSXLNHIK
|
9.7 | IC50 | 4 | — | |
UBWXSCATULGCSA
|
9.7 | IC50 | 4 | — | |
MSOXGTBOMYQLRK
|
9.7 | IC50 | 4 | — | |
WPFZWTKQXNTKQJ
|
9.7 | IC50 | 4 | — | |
KNEKVQSXRQKRBO
|
9.6 | IC50 | 4 | — | |
YWBAOBYDVWSCMN
|
9.6 | IC50 | 4 | — | |
MOWYXIYUNCUBBO
|
9.6 | IC50 | 4 | — | |
FMUGXGTXXNULGS
|
9.6 | IC50 | 4 | — | |
YEQGARBJDLREPV
|
9.5 | IC50 | 4 | — | |
VMQYRLKWZIILQI
|
9.4 | IC50 | 4 | — | |
KITSIKGMHVEYCU
|
9.4 | IC50 | 4 | — | |
NNGVMERLTTVLQP
|
9.3 | IC50 | 8 | — | |
FINZRTUQZUBKBD
|
9.2 | IC50 | 4 | — | |
NQMUJZRUULJLJA
|
9.2 | IC50 | 4 | — | |
FHRWBUZVAOTINV
|
9.2 | IC50 | 4 | — | |
QRYWETQFXDSLKP
|
9.2 | IC50 | 4 | — | |
SUHPRCQYTXOSRF
|
9.1 | IC50 | 4 | — | |
BQFHXEUTDPRCLM
|
9.1 | IC50 | 4 | — | |
LCFFREMLXLZNHE
|
9.1 | IC50 | 5 | — | |
LZOYRTMQLOFTSF
|
9.1 | IC50 | 4 | — | |
GOOMNGHXGYAHJM
|
9.1 | IC50 | 7 | — | |
CYGPGKKCJOVFQJ
|
9.0 | IC50 | 4 | — | |
VJPPLCNBDLZIFG
|
9.0 | IC50 | 5 | — | |
BUXSSQZWDXOIAY
|
9.0 | IC50 | 4 | — | |
IZIBDTDSPVBIEA
|
9.0 | IC50 | 4 | — | |
RXBBNYOZZYEKJZ
|
8.9 | IC50 | 4 | — | |
GFXJEHXKSRGUJJ
|
8.9 | IC50 | 4 | — | |
KKDKMWVZUKAQOJ
|
8.9 | IC50 | 4 | — | |
YFKVYBRENKNUCS
|
8.9 | IC50 | 4 | — | |
ATYAIDXPSYJANV
|
8.9 | IC50 | 4 | — | |
LJODJUIHONTDMR
|
8.9 | IC50 | 7 | — | |
MRGLBSPRZPRKAI
|
8.9 | IC50 | 3 | — | |
STTWMUJSAKOTEV
|
8.9 | IC50 | 4 | — | |
ACWBHJAIEPRBBS
|
8.8 | IC50 | 4 | — | |
JKTAWSRABQDLCF
|
8.8 | IC50 | 4 | — | |
KJRVCMVPIKELBC
|
8.8 | IC50 | 12 | — | |
QLJUTZNCZYGNKW
|
8.8 | IC50 | 4 | — | |
MTQFNASJEDTODL
|
8.8 | IC50 | 4 | — | |
CWBFGXHQESGYOA
|
8.8 | IC50 | 4 | — | |
DEZYACNEATUTOK
|
8.8 | IC50 | 4 | — | |
MPLZFNKPADDSLE
|
8.8 | IC50 | 4 | — |