Target Details
| UniProt AC | P42679 |
|---|---|
| Gene Symbol | MATK |
| Protein Name | Megakaryocyte-associated tyrosine-protein kinase |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07714 (PK_Tyr_Ser-Thr) PF00017 (SH2) PF00018 (SH3_1) |
Summary
- Multi-target molecules 31
- Clinical molecules 3
- Avg pChEMBL 6.46
KEGG Pathways (1)
Active Molecules (31)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
WPHKIQPVPYJNAX
|
7.4 | Ki | 81 | — | |
OWRXHGAFWZFFCW
|
7.3 | Ki | 113 | — | |
MIKAKZKNMYZLDX
|
7.1 | Ki | 42 | — | |
PTSWSUSIGQQZOO
|
7.1 | Ki | 5 | — | |
MZDKLVOWGIOKTN
|
7.0 | Ki | 80 | — | |
RTDSHUGNRVXRHN
|
6.9 | Ki | 51 | — | |
PTVPBWWDGZSEAF
|
6.8 | Ki | 63 | — | |
ZVWRFVCNQOECJS
|
6.8 | Ki | 71 | — | |
GCYXEGSPUDSZJY
|
6.7 | Ki | 82 | — | |
XJSFDMGICAWQFS
|
6.6 | Ki | 60 | — | |
BIIVYFLTOXDAOV
|
6.5 | Ki | 31 | — | |
MVJMMLFMPWITEJ
|
6.5 | Ki | 110 | — | |
VKBFHTIUXUCYRQ
|
6.5 | Ki | 66 | — | |
HKSZLNNOFSGOKW
|
6.4 | IC50 | 408 | — | |
JCFJQIHDZHHMQT
|
6.4 | Ki | 42 | — | |
LYNBNVBMAGDJRW
|
6.4 | Ki | 81 | — | |
XCHWBXBDZRJVDP
|
6.4 | Ki | 51 | — | |
KRIUNPBAQZGFQA
|
6.3 | Ki | 76 | — | |
YMIJUBCSOKSFRU
|
6.3 | Ki | 87 | — | |
PUPCRRRSBUYJAD
|
6.2 | Ki | 44 | Yes | |
RYYNGWLOYLRZLK
|
6.2 | Ki | 104 | — | |
VUHZDNOPEVGHEO
|
6.2 | Ki | 29 | — | |
DZSUJUOJJJCWGG
|
6.1 | Ki | 55 | Yes | |
KJVWCDAPVMWKLJ
|
6.1 | Ki | 20 | — | |
SPYHMOFSJGTUNP
|
6.1 | Ki | 9 | — | |
UIARLYUEJFELEN
|
6.0 | Kd | 289 | Yes | |
BNLPAUPVSCPTDM
|
6.0 | Ki | 15 | — | |
CFIBXVQLBVNOHW
|
6.0 | Ki | 64 | — | |
KWSZYBNXNYRQCC
|
6.0 | Ki | 21 | — | |
ZPXPEKQMLOAPLT
|
6.0 | Ki | 15 | — | |
ZWVZORIKUNOTCS
|
6.0 | Ki | 69 | — |