Target Details
| UniProt AC | P42574 |
|---|---|
| Gene Symbol | CASP3 |
| Protein Name | Caspase-3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00656 (Peptidase_C14) |
Summary
- Multi-target molecules 444
- Clinical molecules 0
- Avg pChEMBL 7.52
KEGG Pathways (46)
- AGE-RAGE signaling pathway in diabetic complications
- Alcoholic liver disease
- Alzheimer disease
- Amoebiasis
- Amyotrophic lateral sclerosis
- Apoptosis
- Apoptosis - multiple species
- Colorectal cancer
- Cytosolic DNA-sensing pathway
- Efferocytosis
- Epithelial cell signaling in Helicobacter pylori infection
- Epstein-Barr virus infection
- Hepatitis B
- Hepatitis C
- Herpes simplex virus 1 infection
- Human cytomegalovirus infection
- Human immunodeficiency virus 1 infection
- Human papillomavirus infection
- Huntington disease
- IL-17 signaling pathway
- Influenza A
- Kaposi sarcoma-associated herpesvirus infection
- Legionellosis
- Lipid and atherosclerosis
- MAPK signaling pathway
- Measles
- MicroRNAs in cancer
- Natural killer cell mediated cytotoxicity
- Non-alcoholic fatty liver disease
- Parkinson disease
- Pathogenic Escherichia coli infection
- Pathways in cancer
- Pathways of neurodegeneration - multiple diseases
- Pertussis
- Platinum drug resistance
- Prion disease
- Proteoglycans in cancer
- Salmonella infection
- Serotonergic synapse
- Small cell lung cancer
- TNF signaling pathway
- Toxoplasmosis
- Tuberculosis
- Viral carcinogenesis
- Viral myocarditis
- p53 signaling pathway
Active Molecules (444)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
YGAZOKVINIORNI
|
6.4 | IC50 | 2 | — | |
LSNJRQWLVIJSDE
|
6.4 | Ki | 3 | — | |
PKCZPKXBVIXOLU
|
6.4 | IC50 | 2 | — | |
RUIXWTIUGYOXFG
|
6.4 | Ki | 3 | — | |
GXKHPUKGZPDYCB
|
6.4 | Ki | 3 | — | |
YZQKWJFJWRAGSA
|
6.4 | IC50 | 2 | — | |
ASGHIPSJIOETFI
|
6.4 | IC50 | 2 | — | |
KNIHFXMFUCCLGH
|
6.4 | IC50 | 5 | — | |
PKQPMQYJGPSJFR
|
6.4 | Ki | 3 | — | |
DOIAAMNEXGWYFQ
|
6.4 | IC50 | 2 | — | |
BILYVLYAAGBKBS
|
6.4 | IC50 | 2 | — | |
AKPWXMAPOSKZGT
|
6.4 | IC50 | 4 | — | |
IMRNKNWXBGSFOO
|
6.4 | IC50 | 2 | — | |
KRXMYBAZKJBJAB
|
6.3 | IC50 | 2 | — | |
NDVYQXXAKHEWLQ
|
6.3 | IC50 | 4 | — | |
YMYGKHWZVMKILN
|
6.3 | IC50 | 2 | — | |
HCWVNDBXTZOJJT
|
6.3 | IC50 | 2 | — | |
HHHCHMWEUVMQER
|
6.3 | IC50 | 4 | — | |
HHHCHMWEUVMQER
|
6.3 | IC50 | 4 | — | |
HIYKUVSVYJWQSQ
|
6.3 | Ki | 3 | — | |
RTXPUAJFUDAYTN
|
6.3 | IC50 | 5 | — | |
WTDVEFVYINBNSI
|
6.3 | Ki | 3 | — | |
KDMQSUUXKLZVNU
|
6.3 | IC50 | 4 | — | |
RTNBVCDVVVYNGZ
|
6.3 | IC50 | 4 | — | |
PBRJUWKZXWXZNB
|
6.3 | IC50 | 2 | — | |
MYQIKQZBTUPQJR
|
6.2 | IC50 | 2 | — | |
JPTDPTOWOMFBRY
|
6.2 | IC50 | 2 | — | |
JPRMMEXMBCGVFV
|
6.1 | IC50 | 2 | — | |
KUYBRHHKOCWADC
|
6.1 | IC50 | 4 | — | |
MEKTUIXWLTWRRE
|
6.1 | IC50 | 4 | — | |
JIFQARCSCBNIIB
|
6.1 | IC50 | 4 | — | |
XDTUFIAIIBWXBZ
|
6.1 | Ki | 3 | — | |
GUHPRPJDBZHYCJ
|
6.1 | IC50 | 3 | — | |
SUUHZYLYARUNIA
|
6.1 | Ki | 3 | — | |
DOBIYIOPZIMMRH
|
6.1 | Ki | 3 | — | |
NERMQYMDDXNPRD
|
6.1 | IC50 | 2 | — | |
KJKPUONOAGOHEL
|
6.0 | Ki | 2 | — | |
VBLKIMKAYGBRKC
|
6.0 | IC50 | 2 | — | |
FUCNIZFCNQFKLX
|
6.0 | IC50 | 2 | — | |
XJQWNXKLHDLZNT
|
6.0 | IC50 | 3 | — | |
KGHGMUBHFANXGE
|
6.0 | IC50 | 2 | — | |
CIDFSOFEWVUWHQ
|
6.0 | IC50 | 4 | — | |
MBJSUONJTWIBKH
|
6.0 | IC50 | 3 | — | |
MBJSUONJTWIBKH
|
6.0 | IC50 | 4 | — |