Target Details
| UniProt AC | P42574 |
|---|---|
| Gene Symbol | CASP3 |
| Protein Name | Caspase-3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00656 (Peptidase_C14) |
Summary
- Multi-target molecules 444
- Clinical molecules 0
- Avg pChEMBL 7.52
KEGG Pathways (46)
- AGE-RAGE signaling pathway in diabetic complications
- Alcoholic liver disease
- Alzheimer disease
- Amoebiasis
- Amyotrophic lateral sclerosis
- Apoptosis
- Apoptosis - multiple species
- Colorectal cancer
- Cytosolic DNA-sensing pathway
- Efferocytosis
- Epithelial cell signaling in Helicobacter pylori infection
- Epstein-Barr virus infection
- Hepatitis B
- Hepatitis C
- Herpes simplex virus 1 infection
- Human cytomegalovirus infection
- Human immunodeficiency virus 1 infection
- Human papillomavirus infection
- Huntington disease
- IL-17 signaling pathway
- Influenza A
- Kaposi sarcoma-associated herpesvirus infection
- Legionellosis
- Lipid and atherosclerosis
- MAPK signaling pathway
- Measles
- MicroRNAs in cancer
- Natural killer cell mediated cytotoxicity
- Non-alcoholic fatty liver disease
- Parkinson disease
- Pathogenic Escherichia coli infection
- Pathways in cancer
- Pathways of neurodegeneration - multiple diseases
- Pertussis
- Platinum drug resistance
- Prion disease
- Proteoglycans in cancer
- Salmonella infection
- Serotonergic synapse
- Small cell lung cancer
- TNF signaling pathway
- Toxoplasmosis
- Tuberculosis
- Viral carcinogenesis
- Viral myocarditis
- p53 signaling pathway
Active Molecules (444)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
KTTPYYAFFJVFFD
|
6.7 | IC50 | 2 | — | |
RBQBJJBLAZNQJZ
|
6.7 | IC50 | 2 | — | |
VCJHWYAJYQWNJL
|
6.7 | IC50 | 2 | — | |
NVEIBIBNNZZXLH
|
6.7 | IC50 | 2 | — | |
PLZURAMCVPIGEB
|
6.7 | IC50 | 2 | — | |
QZDOFOUKELTJRS
|
6.7 | Ki | 3 | — | |
ZUMYWWOOYMHLPE
|
6.7 | IC50 | 2 | — | |
AONGRTQKAZELPJ
|
6.7 | Ki | 2 | — | |
FMTZTJFXNZOBIQ
|
6.7 | Ki | 5 | — | |
QGZFJAMNGXQLQV
|
6.7 | IC50 | 2 | — | |
SHDGJJPFMISTHO
|
6.7 | IC50 | 4 | — | |
XRBANMWDGMCMSJ
|
6.7 | Ki | 3 | — | |
BAOVBFBBIQDDHH
|
6.7 | IC50 | 2 | — | |
WLZOCGMSLPOOIC
|
6.7 | IC50 | 4 | — | |
KQZXEDILUFRWGM
|
6.7 | IC50 | 2 | — | |
NMZRNLRSVKUVJC
|
6.7 | IC50 | 2 | — | |
OBGDVZSRUCWITM
|
6.7 | IC50 | 2 | — | |
QGSAKBWSJFLUIL
|
6.7 | Ki | 3 | — | |
DLYWFYKLKHPATQ
|
6.7 | IC50 | 2 | — | |
GDXMRGIYSQTDEQ
|
6.7 | IC50 | 2 | — | |
IVNMNOZULIYBTB
|
6.6 | IC50 | 2 | — | |
LDDAWLZYJRJPPR
|
6.6 | IC50 | 4 | — | |
QLHHECDAKBHQND
|
6.6 | IC50 | 2 | — | |
CALHLXBTFCJYKI
|
6.6 | IC50 | 2 | — | |
IRZYVIBRQPMBSG
|
6.6 | IC50 | 2 | — | |
QFXLEUGCVOVRCD
|
6.6 | IC50 | 2 | — | |
AHFUCLBQQLXIJB
|
6.6 | Ki | 3 | — | |
GTXNLQVCIHMROL
|
6.6 | IC50 | 2 | — | |
PAPREHNJYFBQSL
|
6.6 | IC50 | 2 | — | |
XXQCRRRNRLLOKC
|
6.6 | IC50 | 2 | — | |
BVAULMYVOSWSBQ
|
6.6 | IC50 | 2 | — | |
QIAVLJUPQMHWEU
|
6.6 | IC50 | 2 | — | |
QIOIIQRMCCDEQM
|
6.6 | IC50 | 2 | — | |
RBQBJJBLAZNQJZ
|
6.6 | IC50 | 2 | — | |
RGINHWLPKMMZFM
|
6.5 | IC50 | 3 | — | |
RGINHWLPKMMZFM
|
6.5 | IC50 | 3 | — | |
KMNYXLBVVHSUPC
|
6.5 | IC50 | 2 | — | |
MIRPJNSLZMOWQE
|
6.5 | IC50 | 2 | — | |
CEFXQYILQBZDCM
|
6.5 | IC50 | 2 | — | |
GQXBVBOSGIYTNU
|
6.5 | IC50 | 2 | — | |
JMCSMHDKXZIFQR
|
6.5 | IC50 | 4 | — | |
FOGVBUNJXCEAOT
|
6.5 | IC50 | 2 | — | |
FGXCHOFOCOXOCJ
|
6.5 | IC50 | 2 | — | |
YYHQMSJBLNLPNZ
|
6.5 | IC50 | 2 | — | |
HOONNWPQCPKYFI
|
6.5 | IC50 | 2 | — | |
HTCDURIAFZLYLG
|
6.5 | Ki | 3 | — | |
LTBPAHIEHDBOIC
|
6.5 | IC50 | 2 | — | |
NCLFPGSWIDLTSV
|
6.5 | IC50 | 2 | — | |
ONFHORMKUAUOAQ
|
6.4 | IC50 | 2 | — | |
XGGOGHVJRTYSOB
|
6.4 | IC50 | 2 | — |