Target Details
| UniProt AC | P42574 |
|---|---|
| Gene Symbol | CASP3 |
| Protein Name | Caspase-3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00656 (Peptidase_C14) |
Summary
- Multi-target molecules 444
- Clinical molecules 0
- Avg pChEMBL 7.52
KEGG Pathways (46)
- AGE-RAGE signaling pathway in diabetic complications
- Alcoholic liver disease
- Alzheimer disease
- Amoebiasis
- Amyotrophic lateral sclerosis
- Apoptosis
- Apoptosis - multiple species
- Colorectal cancer
- Cytosolic DNA-sensing pathway
- Efferocytosis
- Epithelial cell signaling in Helicobacter pylori infection
- Epstein-Barr virus infection
- Hepatitis B
- Hepatitis C
- Herpes simplex virus 1 infection
- Human cytomegalovirus infection
- Human immunodeficiency virus 1 infection
- Human papillomavirus infection
- Huntington disease
- IL-17 signaling pathway
- Influenza A
- Kaposi sarcoma-associated herpesvirus infection
- Legionellosis
- Lipid and atherosclerosis
- MAPK signaling pathway
- Measles
- MicroRNAs in cancer
- Natural killer cell mediated cytotoxicity
- Non-alcoholic fatty liver disease
- Parkinson disease
- Pathogenic Escherichia coli infection
- Pathways in cancer
- Pathways of neurodegeneration - multiple diseases
- Pertussis
- Platinum drug resistance
- Prion disease
- Proteoglycans in cancer
- Salmonella infection
- Serotonergic synapse
- Small cell lung cancer
- TNF signaling pathway
- Toxoplasmosis
- Tuberculosis
- Viral carcinogenesis
- Viral myocarditis
- p53 signaling pathway
Active Molecules (444)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
WTXXKEPFHMWDDX
|
7.0 | IC50 | 2 | — | |
FATMLWUGEBQNST
|
7.0 | IC50 | 2 | — | |
RLJGXAITFUWYPG
|
7.0 | IC50 | 2 | — | |
LBLRFYICWPZBDS
|
7.0 | IC50 | 2 | — | |
SZOQDIPEEPENAN
|
7.0 | Ki | 3 | — | |
IESMBHVLOFERCB
|
7.0 | Ki | 3 | — | |
QMYPHOKIXSLRMB
|
7.0 | IC50 | 2 | — | |
RVUPUUXSFOLOAS
|
7.0 | IC50 | 3 | — | |
QBECUNYDIMMBJO
|
7.0 | Ki | 3 | — | |
VWVKVVPHIDBUPM
|
7.0 | Ki | 3 | — | |
LRVYGOURMARVNX
|
7.0 | Ki | 3 | — | |
RBQBJJBLAZNQJZ
|
7.0 | IC50 | 2 | — | |
NFZRUSZOYOWWEL
|
7.0 | Ki | 3 | — | |
OLSIEGWDJFSEDP
|
7.0 | IC50 | 2 | — | |
CXBBLGYLOAZXJT
|
7.0 | IC50 | 5 | — | |
DIOLAGCWKTXDCP
|
7.0 | IC50 | 2 | — | |
KYGIHIZEIRIHFR
|
7.0 | Ki | 3 | — | |
LNQOGDMGNCKCJV
|
7.0 | IC50 | 2 | — | |
HPLZVLGCPPHPFD
|
6.9 | IC50 | 2 | — | |
DFEUSDFPTOGJKU
|
6.9 | IC50 | 2 | — | |
VUJHWZDCLPHWMO
|
6.9 | Ki | 4 | — | |
CWPCXTXIKFDSTN
|
6.9 | Ki | 3 | — | |
IZSZDPFSJZSGIB
|
6.9 | IC50 | 2 | — | |
SKWCEVYBZPAJGK
|
6.9 | IC50 | 2 | — | |
ZJEAAPUACVGAGQ
|
6.9 | Ki | 3 | — | |
ACQCJOAMWDUQFF
|
6.9 | Ki | 3 | — | |
GBJVAVGBSGRRKN
|
6.9 | IC50 | 2 | — | |
SAUQPQCMYXHHJG
|
6.9 | IC50 | 2 | — | |
PCKDUAQUKNXESJ
|
6.9 | IC50 | 4 | — | |
QVZSKXKXTDTJKH
|
6.9 | IC50 | 2 | — | |
GCIXFQFILPSHQY
|
6.9 | IC50 | 3 | — | |
UVJNVVPTQWFZMT
|
6.9 | IC50 | 4 | — | |
LWBNNPKCSRJWRE
|
6.9 | IC50 | 2 | — | |
NHIDZXMAMOZUNW
|
6.9 | IC50 | 3 | — | |
IBUIGAOZEYCWCZ
|
6.8 | IC50 | 2 | — | |
VMPMJRSSYGKAFD
|
6.8 | IC50 | 2 | — | |
DPMMEOUVESBMSC
|
6.8 | IC50 | 2 | — | |
HVOVPWXTIYQJLM
|
6.8 | Ki | 2 | — | |
HOUWXSCEZSJNPK
|
6.8 | IC50 | 2 | — | |
YIOFGHHAURBGSJ
|
6.8 | IC50 | 3 | — | |
QXPRIMHKXWCGCU
|
6.8 | IC50 | 2 | — | |
DWGRSJBIHVFBFL
|
6.8 | IC50 | 3 | — | |
ABSCBYOPJXYYGS
|
6.8 | Ki | 3 | — | |
VOOBNDVVTJIXRQ
|
6.8 | IC50 | 2 | — | |
AWSNOGJUHYLCCA
|
6.8 | Ki | 3 | — | |
ARFCZUGOPLBBRE
|
6.7 | IC50 | 2 | — | |
KRWGZAGTABTYNO
|
6.7 | IC50 | 3 | — | |
NTFDHIOBCNIACN
|
6.7 | IC50 | 2 | — | |
NVUAKKWTWHVSEV
|
6.7 | IC50 | 2 | — | |
XZTYLVOBUZQRJN
|
6.7 | IC50 | 2 | — |