Target Details
| UniProt AC | P42574 |
|---|---|
| Gene Symbol | CASP3 |
| Protein Name | Caspase-3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00656 (Peptidase_C14) |
Summary
- Multi-target molecules 444
- Clinical molecules 0
- Avg pChEMBL 7.52
KEGG Pathways (46)
- AGE-RAGE signaling pathway in diabetic complications
- Alcoholic liver disease
- Alzheimer disease
- Amoebiasis
- Amyotrophic lateral sclerosis
- Apoptosis
- Apoptosis - multiple species
- Colorectal cancer
- Cytosolic DNA-sensing pathway
- Efferocytosis
- Epithelial cell signaling in Helicobacter pylori infection
- Epstein-Barr virus infection
- Hepatitis B
- Hepatitis C
- Herpes simplex virus 1 infection
- Human cytomegalovirus infection
- Human immunodeficiency virus 1 infection
- Human papillomavirus infection
- Huntington disease
- IL-17 signaling pathway
- Influenza A
- Kaposi sarcoma-associated herpesvirus infection
- Legionellosis
- Lipid and atherosclerosis
- MAPK signaling pathway
- Measles
- MicroRNAs in cancer
- Natural killer cell mediated cytotoxicity
- Non-alcoholic fatty liver disease
- Parkinson disease
- Pathogenic Escherichia coli infection
- Pathways in cancer
- Pathways of neurodegeneration - multiple diseases
- Pertussis
- Platinum drug resistance
- Prion disease
- Proteoglycans in cancer
- Salmonella infection
- Serotonergic synapse
- Small cell lung cancer
- TNF signaling pathway
- Toxoplasmosis
- Tuberculosis
- Viral carcinogenesis
- Viral myocarditis
- p53 signaling pathway
Active Molecules (444)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
IYNNJMRCPJPTMI
|
7.3 | IC50 | 3 | — | |
SLTSJDMMDKNHMN
|
7.3 | Ki | 3 | — | |
WJGNHRNPMJTWAO
|
7.3 | IC50 | 2 | — | |
BEUDVJBODYYMBI
|
7.3 | IC50 | 2 | — | |
NEMHHXQGHOHHKA
|
7.3 | Ki | 3 | — | |
YLVTVASIGAVYHO
|
7.3 | Ki | 3 | — | |
AOUFLZQXBYFGOZ
|
7.3 | IC50 | 3 | — | |
VRYGMTNRJQGMBD
|
7.3 | IC50 | 2 | — | |
JFFCVWIPXCEUGT
|
7.2 | IC50 | 2 | — | |
OEZQRTUGLYPVGI
|
7.2 | IC50 | 2 | — | |
GWEMAMOVSFKYPL
|
7.2 | IC50 | 2 | — | |
GZIHKLOFULVEIA
|
7.2 | Ki | 3 | — | |
JLXZUACSFOZXOH
|
7.2 | IC50 | 2 | — | |
MXGJLIBJKIIQSF
|
7.2 | IC50 | 8 | — | |
GEGJGGLPPHXVSY
|
7.2 | Ki | 3 | — | |
WIYBIQZLIVGWQF
|
7.2 | IC50 | 3 | — | |
ZQDAIIUFJKGWON
|
7.2 | IC50 | 2 | — | |
ACPNTFIHYLLTHQ
|
7.2 | IC50 | 2 | — | |
DCKBIXRXOAUIHS
|
7.2 | Ki | 3 | — | |
FZIXMTMBUYOGCV
|
7.2 | IC50 | 2 | — | |
IPHOHJYEJYKOEY
|
7.2 | IC50 | 2 | — | |
KTOSNSDXQPHMPE
|
7.2 | Ki | 3 | — | |
CSUJUVXXFCVRHL
|
7.2 | Ki | 3 | — | |
DPRGPUSLFXWJTI
|
7.2 | Ki | 3 | — | |
CRXIPRWVEVJYQK
|
7.2 | Ki | 3 | — | |
YERUFWIDABDQJG
|
7.2 | Ki | 3 | — | |
ACJYSQZZDDSVHX
|
7.2 | Ki | 3 | — | |
YNDYWRFJZGWCJS
|
7.2 | IC50 | 2 | — | |
DZHQUOCAZBRQCK
|
7.2 | Ki | 3 | — | |
RZIOHTDLDUFVCW
|
7.2 | IC50 | 4 | — | |
VSSIZIZQEBJUBI
|
7.2 | Ki | 3 | — | |
MZDVCOYYTAHLOR
|
7.2 | Ki | 3 | — | |
USLSSPUBZCKDRS
|
7.2 | Ki | 3 | — | |
AAGJQHMOJORKRA
|
7.1 | IC50 | 2 | — | |
IDXGNHSBSFGHCS
|
7.1 | IC50 | 2 | — | |
VMHZRSKJCWWRNQ
|
7.1 | IC50 | 2 | — | |
BVPRPKGQOIQLMI
|
7.1 | IC50 | 2 | — | |
NKXHLTPOYVGFQY
|
7.1 | Ki | 3 | — | |
DPNDRYUDIJORHR
|
7.1 | IC50 | 2 | — | |
KYUFGGNCJRWMDN
|
7.1 | IC50 | 5 | — | |
IRBBDJYBNHNLKO
|
7.1 | IC50 | 2 | — | |
YGIPKOMPEBEYJK
|
7.1 | IC50 | 2 | — | |
ZQZYDAYNBPNRDV
|
7.1 | IC50 | 2 | — | |
FNPIWKPAAMBRAA
|
7.1 | IC50 | 2 | — | |
JMIGYLZAZILEMQ
|
7.1 | Ki | 3 | — | |
KECFNHULKQPLHJ
|
7.1 | IC50 | 2 | — | |
XNELIBGPKZNEOG
|
7.1 | IC50 | 5 | — | |
SLQMNVJNDYLJSF
|
7.1 | IC50 | 2 | — | |
MIQOWTZVMDSHBY
|
7.1 | IC50 | 2 | — | |
FIEQQFOHZKVJLV
|
7.0 | Ki | 2 | — |