Target Details
| UniProt AC | P42574 |
|---|---|
| Gene Symbol | CASP3 |
| Protein Name | Caspase-3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00656 (Peptidase_C14) |
Summary
- Multi-target molecules 444
- Clinical molecules 0
- Avg pChEMBL 7.52
KEGG Pathways (46)
- AGE-RAGE signaling pathway in diabetic complications
- Alcoholic liver disease
- Alzheimer disease
- Amoebiasis
- Amyotrophic lateral sclerosis
- Apoptosis
- Apoptosis - multiple species
- Colorectal cancer
- Cytosolic DNA-sensing pathway
- Efferocytosis
- Epithelial cell signaling in Helicobacter pylori infection
- Epstein-Barr virus infection
- Hepatitis B
- Hepatitis C
- Herpes simplex virus 1 infection
- Human cytomegalovirus infection
- Human immunodeficiency virus 1 infection
- Human papillomavirus infection
- Huntington disease
- IL-17 signaling pathway
- Influenza A
- Kaposi sarcoma-associated herpesvirus infection
- Legionellosis
- Lipid and atherosclerosis
- MAPK signaling pathway
- Measles
- MicroRNAs in cancer
- Natural killer cell mediated cytotoxicity
- Non-alcoholic fatty liver disease
- Parkinson disease
- Pathogenic Escherichia coli infection
- Pathways in cancer
- Pathways of neurodegeneration - multiple diseases
- Pertussis
- Platinum drug resistance
- Prion disease
- Proteoglycans in cancer
- Salmonella infection
- Serotonergic synapse
- Small cell lung cancer
- TNF signaling pathway
- Toxoplasmosis
- Tuberculosis
- Viral carcinogenesis
- Viral myocarditis
- p53 signaling pathway
Active Molecules (444)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
HWKXAKRQXXUBFD
|
7.5 | IC50 | 3 | — | |
HWKXAKRQXXUBFD
|
7.5 | IC50 | 3 | — | |
VUTPSTRRGSVYGS
|
7.5 | Ki | 3 | — | |
RYWKNTKVPRMYNJ
|
7.5 | IC50 | 2 | — | |
AYQUXMOMSNPZEF
|
7.5 | Ki | 4 | — | |
HIQKYBKHPZKDSE
|
7.5 | IC50 | 2 | — | |
LYBWGROBJJXCJJ
|
7.5 | IC50 | 6 | — | |
SIHWSNWMVORLAP
|
7.5 | IC50 | 2 | — | |
UPNDCXMMARFRPM
|
7.5 | IC50 | 3 | — | |
URMGPEOQLIISAB
|
7.5 | Ki | 4 | — | |
VCWYKJKQZUPTQP
|
7.5 | Ki | 2 | — | |
XTKUMMDOZMHSCM
|
7.5 | IC50 | 2 | — | |
YPVHLSJXDPMUQA
|
7.5 | IC50 | 5 | — | |
GIUGBCHQBCYCTJ
|
7.5 | IC50 | 2 | — | |
UMHSZDAKIVGDNR
|
7.5 | IC50 | 3 | — | |
UZQYVRYDJUXDFW
|
7.5 | IC50 | 2 | — | |
DCOFJYKNJPKGOK
|
7.5 | Ki | 3 | — | |
JEYQBANFJYIELI
|
7.5 | IC50 | 4 | — | |
LHHQIZSDNGIYTJ
|
7.5 | IC50 | 2 | — | |
CJCQGCDZQWKTQF
|
7.5 | IC50 | 2 | — | |
RQWMOUMJTFUKRW
|
7.5 | IC50 | 2 | — | |
SIQQBFWEHZXLAO
|
7.5 | IC50 | 6 | — | |
ZDXBUNGSLQDEGV
|
7.5 | IC50 | 2 | — | |
TXWGTLBORQHCEB
|
7.5 | IC50 | 2 | — | |
VJNOWWSHWOXTFM
|
7.5 | Ki | 3 | — | |
WWBXAIBXPFRZEI
|
7.5 | Ki | 3 | — | |
JYCOKQSQAYKENG
|
7.4 | Ki | 3 | — | |
RZTNFNUQIOVICT
|
7.4 | Ki | 3 | — | |
NKBDSMREMMRFSI
|
7.4 | IC50 | 5 | — | |
NKBDSMREMMRFSI
|
7.4 | IC50 | 5 | — | |
PZMBYHSWPUMKMR
|
7.4 | Ki | 3 | — | |
VFANYHPZKZVWGL
|
7.4 | IC50 | 2 | — | |
ACIRQJGPTIFUPJ
|
7.4 | IC50 | 2 | — | |
PIQHWGFQAFGKBN
|
7.4 | IC50 | 2 | — | |
ZHCWWOOIEILUBJ
|
7.4 | Ki | 3 | — | |
HIAYBHWMULSKJU
|
7.4 | Ki | 3 | — | |
MAMIJEIFDIXCPX
|
7.4 | Ki | 4 | — | |
OYAQGPKREWSCAC
|
7.4 | Ki | 3 | — | |
ULPLTJMGFAFYSR
|
7.4 | IC50 | 2 | — | |
FGBBQLKNFNUJTG
|
7.4 | IC50 | 2 | — | |
GOKIOWHGQQDARQ
|
7.4 | Ki | 3 | — | |
QIZVTMONNDOOLR
|
7.4 | IC50 | 2 | — | |
WAEPNLVCPPIQJQ
|
7.4 | Ki | 3 | — | |
QKVWMYQCBWNCQH
|
7.4 | IC50 | 2 | — | |
QERRYNKMJLOQEN
|
7.3 | Ki | 3 | — | |
VMDJSHWGYGBHNX
|
7.3 | Ki | 3 | — | |
AJJFEZDYZOETDJ
|
7.3 | IC50 | 2 | — | |
RSWZABGNSYHJJL
|
7.3 | IC50 | 2 | — | |
SDEQMNUREZLDJE
|
7.3 | IC50 | 2 | — | |
BZEURKGKCWHMON
|
7.3 | Ki | 4 | — |