Target Details
| UniProt AC | P42574 |
|---|---|
| Gene Symbol | CASP3 |
| Protein Name | Caspase-3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00656 (Peptidase_C14) |
Summary
- Multi-target molecules 444
- Clinical molecules 0
- Avg pChEMBL 7.52
KEGG Pathways (46)
- AGE-RAGE signaling pathway in diabetic complications
- Alcoholic liver disease
- Alzheimer disease
- Amoebiasis
- Amyotrophic lateral sclerosis
- Apoptosis
- Apoptosis - multiple species
- Colorectal cancer
- Cytosolic DNA-sensing pathway
- Efferocytosis
- Epithelial cell signaling in Helicobacter pylori infection
- Epstein-Barr virus infection
- Hepatitis B
- Hepatitis C
- Herpes simplex virus 1 infection
- Human cytomegalovirus infection
- Human immunodeficiency virus 1 infection
- Human papillomavirus infection
- Huntington disease
- IL-17 signaling pathway
- Influenza A
- Kaposi sarcoma-associated herpesvirus infection
- Legionellosis
- Lipid and atherosclerosis
- MAPK signaling pathway
- Measles
- MicroRNAs in cancer
- Natural killer cell mediated cytotoxicity
- Non-alcoholic fatty liver disease
- Parkinson disease
- Pathogenic Escherichia coli infection
- Pathways in cancer
- Pathways of neurodegeneration - multiple diseases
- Pertussis
- Platinum drug resistance
- Prion disease
- Proteoglycans in cancer
- Salmonella infection
- Serotonergic synapse
- Small cell lung cancer
- TNF signaling pathway
- Toxoplasmosis
- Tuberculosis
- Viral carcinogenesis
- Viral myocarditis
- p53 signaling pathway
Active Molecules (444)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
COLCPJSXGNKCEG
|
8.1 | IC50 | 2 | — | |
FNURIBXCMKMVRL
|
8.0 | IC50 | 2 | — | |
GCQVILHNVZSRTL
|
8.0 | IC50 | 2 | — | |
IXNAXPALFGYLBG
|
8.0 | IC50 | 2 | — | |
VZUJUIONFIJSIE
|
8.0 | IC50 | 3 | — | |
JPCVJWQLKRHLRX
|
8.0 | IC50 | 3 | — | |
JRPNHUJRYWPJMH
|
8.0 | IC50 | 2 | — | |
JVKBLHAUEXSZHN
|
8.0 | IC50 | 2 | — | |
WXJHOKNCTBSTEM
|
8.0 | IC50 | 2 | — | |
CUDGJBLALZRKFR
|
8.0 | IC50 | 3 | — | |
FZAVLWDWOZHIBJ
|
8.0 | IC50 | 3 | — | |
MFHQDLHNUMVDLA
|
8.0 | IC50 | 4 | — | |
OJYJCHGYJSCGSY
|
8.0 | IC50 | 2 | — | |
SGVNFLQYMIJSSK
|
8.0 | IC50 | 3 | — | |
MSJFYYXGZZIVOJ
|
8.0 | IC50 | 2 | — | |
KYJSQQPQAAKFQY
|
8.0 | IC50 | 2 | — | |
RVXFIJCZJQLWSY
|
8.0 | IC50 | 2 | — | |
SVBRVLOFXVNEPG
|
8.0 | IC50 | 2 | — | |
UITSDZFHHJSHNP
|
8.0 | IC50 | 2 | — | |
XXUBHIOESHILCG
|
8.0 | IC50 | 2 | — | |
IEGXKLYPPWABDL
|
8.0 | IC50 | 2 | — | |
CGZTYJDMCMAZBO
|
7.9 | IC50 | 2 | — | |
CXJCEKSGEFHWMX
|
7.9 | IC50 | 2 | — | |
RBCPNDRFXKBOQT
|
7.9 | IC50 | 2 | — | |
BLQICVVKCWCIMT
|
7.9 | IC50 | 2 | — | |
BSDZXTVQJICEPK
|
7.9 | IC50 | 2 | — | |
OEZQRTUGLYPVGI
|
7.9 | IC50 | 2 | — | |
RGKPGQYSJPTIFN
|
7.9 | IC50 | 2 | — | |
RRBOQMCBPIXZCY
|
7.9 | IC50 | 2 | — | |
SNETYMFZDXAJJJ
|
7.9 | IC50 | 2 | — | |
STDJONDOUCKJSO
|
7.9 | IC50 | 3 | — | |
STDJONDOUCKJSO
|
7.9 | IC50 | 3 | — | |
PKOUAUWPBMZQCH
|
7.9 | IC50 | 3 | — | |
ZJPAUGHACIPCFI
|
7.9 | IC50 | 2 | — | |
FOBVNTSMOHZMIV
|
7.9 | Ki | 3 | — | |
NUEXSSWTCJYNJY
|
7.9 | IC50 | 4 | — | |
UUXBTSRITCUIRR
|
7.9 | IC50 | 4 | — | |
VMCLZBMIORMDHX
|
7.9 | Ki | 3 | — | |
ZSLCIFACVMMVCF
|
7.9 | IC50 | 2 | — | |
WWOJLWFIFRTCON
|
7.9 | IC50 | 2 | — | |
IPBPQSZVGDLNHE
|
7.9 | IC50 | 2 | — | |
DKRXATGOSDBMOO
|
7.9 | IC50 | 2 | — | |
HBEKNGSODXFMMQ
|
7.9 | IC50 | 2 | — | |
ULYGADBUPXIMGK
|
7.9 | IC50 | 2 | — | |
XBDITFWCQVJBBF
|
7.9 | IC50 | 2 | — | |
HYYDYCCTMBTVAC
|
7.8 | IC50 | 2 | — | |
PTQPGYBOZKMKKV
|
7.8 | Ki | 3 | — | |
YSDNTHYUFYFOEN
|
7.8 | IC50 | 4 | — | |
AMNQDPUKNDHUGB
|
7.8 | IC50 | 2 | — | |
GKHVWLIRHANJNR
|
7.8 | Ki | 3 | — |