Target Details
| UniProt AC | P42574 |
|---|---|
| Gene Symbol | CASP3 |
| Protein Name | Caspase-3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00656 (Peptidase_C14) |
Summary
- Multi-target molecules 444
- Clinical molecules 0
- Avg pChEMBL 7.52
KEGG Pathways (46)
- AGE-RAGE signaling pathway in diabetic complications
- Alcoholic liver disease
- Alzheimer disease
- Amoebiasis
- Amyotrophic lateral sclerosis
- Apoptosis
- Apoptosis - multiple species
- Colorectal cancer
- Cytosolic DNA-sensing pathway
- Efferocytosis
- Epithelial cell signaling in Helicobacter pylori infection
- Epstein-Barr virus infection
- Hepatitis B
- Hepatitis C
- Herpes simplex virus 1 infection
- Human cytomegalovirus infection
- Human immunodeficiency virus 1 infection
- Human papillomavirus infection
- Huntington disease
- IL-17 signaling pathway
- Influenza A
- Kaposi sarcoma-associated herpesvirus infection
- Legionellosis
- Lipid and atherosclerosis
- MAPK signaling pathway
- Measles
- MicroRNAs in cancer
- Natural killer cell mediated cytotoxicity
- Non-alcoholic fatty liver disease
- Parkinson disease
- Pathogenic Escherichia coli infection
- Pathways in cancer
- Pathways of neurodegeneration - multiple diseases
- Pertussis
- Platinum drug resistance
- Prion disease
- Proteoglycans in cancer
- Salmonella infection
- Serotonergic synapse
- Small cell lung cancer
- TNF signaling pathway
- Toxoplasmosis
- Tuberculosis
- Viral carcinogenesis
- Viral myocarditis
- p53 signaling pathway
Active Molecules (444)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
SCZQZYJOIBQIGS
|
8.6 | IC50 | 4 | — | |
DOVOIZGMETXBAW
|
8.5 | IC50 | 2 | — | |
OYEOXFZRVNDRKZ
|
8.5 | IC50 | 5 | — | |
ABCKZNSVBLCRMS
|
8.5 | IC50 | 3 | — | |
IYOWHFAECQXBOU
|
8.5 | IC50 | 2 | — | |
UMBVAPCONCILTL
|
8.5 | IC50 | 5 | — | |
IYUHLZOWOKCWMK
|
8.5 | IC50 | 3 | — | |
YDPWIEQYFRHMKK
|
8.5 | IC50 | 2 | — | |
INEQQSYFBJJTKI
|
8.5 | IC50 | 5 | — | |
ZFUKMGBZRXETJQ
|
8.5 | IC50 | 3 | — | |
APKUVGMUIXJJAR
|
8.4 | IC50 | 2 | — | |
YYTCWUDLORCZAE
|
8.4 | IC50 | 2 | — | |
ZUPAARUJOOKFLI
|
8.4 | IC50 | 2 | — | |
CLKQXEGDLZQTME
|
8.4 | IC50 | 4 | — | |
MPIKODMIUDLWKY
|
8.4 | IC50 | 3 | — | |
OCRBUZYTFNEEGD
|
8.4 | IC50 | 2 | — | |
XDHJBIYJRNFDKS
|
8.4 | IC50 | 2 | — | |
IZQMNYSMAWSYDA
|
8.4 | IC50 | 2 | — | |
YIXFIKCRDGRBDB
|
8.4 | IC50 | 2 | — | |
BTAFTKGHXXQLHC
|
8.3 | IC50 | 4 | — | |
SDUIHZXGXLYNPJ
|
8.3 | IC50 | 2 | — | |
XUUQUFQWQGVYPU
|
8.3 | IC50 | 2 | — | |
AEYFPXLRNOQPNR
|
8.3 | IC50 | 2 | — | |
FLSOPDBNBOFSSL
|
8.3 | IC50 | 2 | — | |
NKBSCZIQSOVWKJ
|
8.3 | IC50 | 3 | — | |
NKBSCZIQSOVWKJ
|
8.3 | IC50 | 3 | — | |
NQNOSUGXDKSHRE
|
8.3 | IC50 | 3 | — | |
PSEYKDQFSOGYNR
|
8.3 | IC50 | 4 | — | |
QENZECCKNUZHEO
|
8.3 | IC50 | 3 | — | |
VIKAKOARTUQKPC
|
8.3 | IC50 | 3 | — | |
XIMITGPWYYFUQF
|
8.3 | Ki | 5 | — | |
FXRYYTKWISSZGE
|
8.3 | IC50 | 2 | — | |
PCWDXECMTMSSCD
|
8.3 | IC50 | 2 | — | |
QGTNZCUWEMSWQW
|
8.2 | IC50 | 2 | — | |
CHBXPPLGXKEWKQ
|
8.2 | IC50 | 2 | — | |
WZRDTXYFPUFFST
|
8.2 | IC50 | 3 | — | |
XIMITGPWYYFUQF
|
8.2 | IC50 | 3 | — | |
GAHXAXBPTNBDFH
|
8.2 | IC50 | 2 | — | |
XKFNXVGANVXVEU
|
8.2 | IC50 | 2 | — | |
AEVFCJHPCHDXDJ
|
8.2 | IC50 | 2 | — | |
UUEMWRIOZLIPHU
|
8.2 | IC50 | 4 | — | |
UUEMWRIOZLIPHU
|
8.2 | IC50 | 4 | — | |
BPUYCCMTBNUYAN
|
8.2 | IC50 | 2 | — | |
BBHZJDWNUYJWFP
|
8.1 | IC50 | 2 | — | |
JQQCMQLLJHRXIA
|
8.1 | IC50 | 2 | — | |
IFZWBMQGMKRQEH
|
8.1 | IC50 | 2 | — | |
LPQXQLRRATZAID
|
8.1 | IC50 | 2 | — | |
MBFCFVOWKKZRNA
|
8.1 | IC50 | 2 | — | |
TYGQNSUHNPKJOA
|
8.1 | IC50 | 2 | — | |
QCKJEQIYOITZDI
|
8.1 | IC50 | 2 | — |