Target Details
| UniProt AC | P42574 |
|---|---|
| Gene Symbol | CASP3 |
| Protein Name | Caspase-3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00656 (Peptidase_C14) |
Summary
- Multi-target molecules 444
- Clinical molecules 0
- Avg pChEMBL 7.52
KEGG Pathways (46)
- AGE-RAGE signaling pathway in diabetic complications
- Alcoholic liver disease
- Alzheimer disease
- Amoebiasis
- Amyotrophic lateral sclerosis
- Apoptosis
- Apoptosis - multiple species
- Colorectal cancer
- Cytosolic DNA-sensing pathway
- Efferocytosis
- Epithelial cell signaling in Helicobacter pylori infection
- Epstein-Barr virus infection
- Hepatitis B
- Hepatitis C
- Herpes simplex virus 1 infection
- Human cytomegalovirus infection
- Human immunodeficiency virus 1 infection
- Human papillomavirus infection
- Huntington disease
- IL-17 signaling pathway
- Influenza A
- Kaposi sarcoma-associated herpesvirus infection
- Legionellosis
- Lipid and atherosclerosis
- MAPK signaling pathway
- Measles
- MicroRNAs in cancer
- Natural killer cell mediated cytotoxicity
- Non-alcoholic fatty liver disease
- Parkinson disease
- Pathogenic Escherichia coli infection
- Pathways in cancer
- Pathways of neurodegeneration - multiple diseases
- Pertussis
- Platinum drug resistance
- Prion disease
- Proteoglycans in cancer
- Salmonella infection
- Serotonergic synapse
- Small cell lung cancer
- TNF signaling pathway
- Toxoplasmosis
- Tuberculosis
- Viral carcinogenesis
- Viral myocarditis
- p53 signaling pathway
Active Molecules (444)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
YNRQFMSSDVQNGQ
|
11.8 | Ki | 8 | — | |
CKRCPAGGKUFVIT
|
11.5 | IC50 | 4 | — | |
XIMITGPWYYFUQF
|
11.3 | Ki | 8 | — | |
XWTJWAAMOCNKHH
|
11.0 | IC50 | 4 | — | |
JYGKCHPWCXRSQJ
|
9.8 | IC50 | 4 | — | |
QFAGZHXWKDBXGQ
|
9.7 | IC50 | 4 | — | |
SFDIMTVHWVLTIP
|
9.7 | IC50 | 4 | — | |
ULELQXPHOSNTHT
|
9.6 | IC50 | 4 | — | |
UCOGGEXRPKAPHO
|
9.6 | IC50 | 3 | — | |
GQDJBEWJIKPEQS
|
9.5 | IC50 | 3 | — | |
MBPKVWLXSMFUMN
|
9.4 | IC50 | 4 | — | |
GGRODTCKLDDOBP
|
9.4 | IC50 | 3 | — | |
MDRQEFUKIMUQFX
|
9.4 | IC50 | 4 | — | |
QAFBFHNIUINEJN
|
9.4 | IC50 | 4 | — | |
HDXDXAKYCMKPSF
|
9.3 | IC50 | 4 | — | |
INTJRTIYLCEHRJ
|
9.3 | IC50 | 4 | — | |
CSEDBYKWGJUWMQ
|
9.3 | IC50 | 3 | — | |
MTGSTDMYYFQKEE
|
9.3 | IC50 | 3 | — | |
SVQAMGNGTJSUFV
|
9.3 | IC50 | 3 | — | |
GCDOZFZRBUNMDE
|
9.2 | IC50 | 3 | — | |
NJAQASWTRGUAGC
|
9.2 | IC50 | 3 | — | |
NHHJXCJHJPGPEF
|
9.1 | IC50 | 4 | — | |
LVXZMAMJNHAXKU
|
9.1 | IC50 | 4 | — | |
MNAXVQLJZGETJF
|
9.1 | IC50 | 3 | — | |
OOGHGBCRVSBUHH
|
9.0 | Ki | 3 | — | |
ZXYUJUZVJDHMDR
|
9.0 | IC50 | 4 | — | |
DONUNLOVYIQJNS
|
8.9 | IC50 | 4 | — | |
VXDALODUEXZZKU
|
8.9 | IC50 | 2 | — | |
XIMSCIZHMWOJHC
|
8.9 | IC50 | 3 | — | |
YNRQFMSSDVQNGQ
|
8.8 | Ki | 5 | — | |
QLHDEYZCVHOGEF
|
8.8 | IC50 | 4 | — | |
NAZSWKZWCFVHEL
|
8.8 | IC50 | 4 | — | |
GEZSSSVQIGDDMR
|
8.8 | IC50 | 4 | — | |
KSIBLECLZAACGQ
|
8.8 | IC50 | 3 | — | |
OOMWRPAWHLYIEI
|
8.8 | IC50 | 2 | — | |
UWYWIWOJPZFFAT
|
8.8 | IC50 | 4 | — | |
OMCJYUDICKFVIV
|
8.7 | IC50 | 2 | — | |
NCCIOJYCWRHZMY
|
8.7 | IC50 | 4 | — | |
SHHIOGGLCRQOHT
|
8.7 | IC50 | 4 | — | |
SKSZJGAFHISZNB
|
8.7 | IC50 | 5 | — | |
HIBILFREOVFCHQ
|
8.7 | IC50 | 4 | — | |
NETBIBQTHPVZHP
|
8.6 | IC50 | 4 | — | |
VBXOCZFAWPHIJQ
|
8.6 | IC50 | 3 | — | |
XBILASWQSBQTIV
|
8.6 | IC50 | 2 | — | |
SMINLRKVPPXJGK
|
8.6 | IC50 | 2 | — | |
BPPAKSZSGBPOEH
|
8.6 | IC50 | 4 | — | |
UUTWTWROPLXGDT
|
8.6 | IC50 | 3 | — | |
RIBWEGLQTVTLTI
|
8.6 | IC50 | 2 | — | |
WPBCCSIRQOJBIN
|
8.6 | IC50 | 3 | — | |
LQXYDGHSLQNYCW
|
8.6 | IC50 | 2 | — |