Target Details
| UniProt AC | P42356 |
|---|---|
| Gene Symbol | PI4KA |
| Protein Name | Phosphatidylinositol 4-kinase alpha |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00454 (PI3_PI4_kinase) PF00613 (PI3Ka) PF19274 (PI4K_N) |
Summary
- Multi-target molecules 41
- Clinical molecules 1
- Avg pChEMBL 7.29
KEGG Pathways (3)
Associated Diseases (3)
Active Molecules (41)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
LEPAEWXGTXYMEY
|
9.5 | IC50 | 2 | — | |
DSQJVZCCWLGHTH
|
9.0 | IC50 | 2 | — | |
FEXTUSFUMVYBFH
|
9.0 | IC50 | 2 | — | |
LCUPEZBPGVQFLN
|
9.0 | IC50 | 2 | — | |
BITYGNDFPWCLCP
|
8.8 | IC50 | 2 | — | |
XHJVXWBRJUGTON
|
8.8 | IC50 | 2 | — | |
WYCWXWHOPSRYNV
|
8.7 | IC50 | 2 | — | |
JLAZWUFUZDVBSK
|
8.4 | IC50 | 2 | — | |
FEUPFWSRAMSZRO
|
8.3 | IC50 | 2 | — | |
JBMPVRPUGHDUOL
|
8.3 | IC50 | 2 | — | |
WTFBXXYMHMHBJI
|
8.1 | IC50 | 2 | — | |
BTUKQVYIQOODQH
|
8.0 | IC50 | 2 | — | |
HSNVRQXJCBRZAG
|
8.0 | IC50 | 2 | — | |
CVFBATDOQSKZOU
|
7.7 | IC50 | 2 | — | |
QQCJQRGQHJYFGI
|
7.5 | IC50 | 2 | — | |
FFFQPROXASWICG
|
7.4 | IC50 | 2 | — | |
FKUAUADTVPZXDK
|
7.4 | IC50 | 2 | — | |
KJVHQZBJZUVKEB
|
7.3 | IC50 | 2 | — | |
ISKUKBKBISOCEK
|
7.0 | IC50 | 2 | — | |
PPECOBBFKIXTSR
|
7.0 | IC50 | 3 | — | |
XMKQZYFAHHTULJ
|
6.9 | IC50 | 2 | — | |
BRHYDYVHLAHDCZ
|
6.9 | IC50 | 7 | — | |
BYTQGWNNPKNUGP
|
6.8 | IC50 | 2 | — | |
VNQBKUWYQVWGPY
|
6.8 | IC50 | 2 | — | |
VKOFOXNLTIKFHE
|
6.8 | IC50 | 8 | — | |
IHWSJFBJORCEAK
|
6.8 | IC50 | 7 | — | |
QDLHCMPXEPAAMD
|
6.5 | IC50 | 13 | Yes | |
CJLFOZCDDFNSOD
|
6.5 | IC50 | 2 | — | |
QIVYBELVULYGBM
|
6.5 | IC50 | 2 | — | |
VFAOZGIUZWPHKS
|
6.5 | IC50 | 2 | — | |
VWBMWDWXMHMJPH
|
6.5 | IC50 | 2 | — | |
YUTIPCGWKBPNFQ
|
6.5 | IC50 | 2 | — | |
KCZKGYFLHBVLMU
|
6.4 | IC50 | 5 | — | |
GKHVKQHALKASHA
|
6.3 | IC50 | 2 | — | |
ZOCGDBROXGJXNN
|
6.3 | IC50 | 2 | — | |
PIBKKQFQADCDAW
|
6.2 | IC50 | 7 | — | |
CBBGVZCNBLEQID
|
6.2 | IC50 | 5 | — | |
IPLZEFLYSZCVED
|
6.2 | IC50 | 2 | — | |
HORACVGDHNAIMC
|
6.2 | IC50 | 2 | — | |
PGBDHJBYFJSWIV
|
6.0 | IC50 | 2 | — | |
ZYCQTLJPCIVXNL
|
6.0 | IC50 | 4 | — |