Target Details
UniProt ACP42336
Gene SymbolPIK3CA
Protein NamePhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00454 (PI3_PI4_kinase) PF00792 (PI3K_C2) PF02192 (PI3K_p85B) PF00794 (PI3K_rbd) PF00613 (PI3Ka)
Summary
  • Multi-target molecules 5,616
  • Clinical molecules 115
  • Avg pChEMBL 7.53
KEGG Pathways (109)
Top Co-occurrence Targets
Active Molecules (5,616)
InChIKey pChEMBL Type Targets Clinical
LONMISVNAYVDGX 11.0 Ki 2
ROYQBLPXACEGTQ 10.8 Ki 2
GEUADBGMXZNPKD 10.8 Ki 2
HABOHZQRJSLFDW 10.7 Ki 2
KFPLPXINZUQEEC 10.7 Ki 2
QDEYUYMESVXMGP 10.7 Ki 2
YNKNMRFZPSXUSI 10.7 Ki 2
LIDOSBIJMNIHPF 10.7 Ki 2
AOSWTRNJUDHHEV 10.7 Ki 2
FXNPXFSTJWGUJP 10.7 Ki 2
MPJAHOIDOOABIN 10.7 Ki 2
ODACICVNFSDKGJ 10.7 Ki 2
GEUADBGMXZNPKD 10.7 Ki 2
GYTQULHCMOEAHF 10.7 Ki 2
HJKORHLOCBIOOW 10.7 Ki 2
ILXAWHFQWWTBNG 10.7 Ki 4
OBBDENVJGIGQIP 10.7 Ki 2
QAAIJJGWIRSNIR 10.7 Ki 2
YSHXJRZRFDGXCH 10.7 Ki 2
AHNACMAJVLLNSG 10.6 Ki 4
MMDOIDWSYTUJEP 10.6 Ki 2
NAPNAGZGKVCYGY 10.6 Ki 4
BEYUPKZHHDIWGS 10.6 Ki 2
CLFAMUPHBRSLEU 10.6 Ki 2
DJXUVDUIQQGXRO 10.6 Ki 2
IWTPWLVQNOYAOH 10.6 Ki 2
QQCCDSJWSBTDAK 10.6 Ki 2
QVSZGFWEMFZULG 10.6 Ki 2
YIKWEFOKXWDICJ 10.6 Ki 2
QYTPRNFXBNNVPK 10.6 Ki 2
ROLFNMFERWVMML 10.6 Ki 2
WCCXUZJXPGCBTF 10.6 Ki 2
CQUHGORAXVYLJW 10.6 Ki 2
FNEUXHRPWFQLDN 10.6 Ki 2
MNSXRVQYVXOLAY 10.6 Ki 2
ONIMSHRZEOOAPG 10.6 Ki 2
VKHJFKVLUCPKMG 10.6 Ki 2
WBTZQNMPEFHDOP 10.6 Ki 2
XEQUZSZPETWUBR 10.6 Ki 2
BFYFVGVWNGHSAB 10.6 Ki 2
LRDXLDYDJFBFCE 10.6 Ki 2
SRJXASRLXDINEX 10.6 Ki 2
SZAXYAOPUVXVDN 10.6 Ki 2
TXIVOMAGVACXTL 10.6 Ki 2
ZXKOCPUQTKZNJM 10.6 Ki 2
LBAUYAOVGJAFQD 10.6 Ki 2
LRDXLDYDJFBFCE 10.6 Ki 2
AYKSFHQCPBPUPW 10.5 Ki 2
ZLADDXGUXPSLGC 10.5 Ki 2
BFXVGQSVKWTOAL 10.5 Ki 2
2D structure