Target Details
| UniProt AC | P42261 |
|---|---|
| Gene Symbol | GRIA1 |
| Protein Name | Glutamate receptor 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF01094 (ANF_receptor) PF00060 (Lig_chan) PF10613 (Lig_chan-Glu_bd) |
Summary
- Multi-target molecules 143
- Clinical molecules 0
- Avg pChEMBL 7.18
KEGG Pathways (15)
- Amphetamine addiction
- Amyotrophic lateral sclerosis
- Circadian entrainment
- Dopaminergic synapse
- Glutamatergic synapse
- Huntington disease
- Long-term depression
- Long-term potentiation
- Neuroactive ligand signaling
- Neuroactive ligand-receptor interaction
- Nicotine addiction
- Pathways of neurodegeneration - multiple diseases
- Retrograde endocannabinoid signaling
- Spinocerebellar ataxia
- cAMP signaling pathway
Associated Diseases (2)
Active Molecules (143)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
JASCMFDYTJFEAR
|
6.6 | IC50 | 4 | — | |
CVQAHSMQXIWVLD
|
6.6 | Ki | 4 | — | |
IEBVITXSHAFLJR
|
6.5 | Ki | 4 | — | |
RWVIMCIPOAXUDG
|
6.5 | IC50 | 11 | — | |
UCTNZJNATOCSCH
|
6.5 | Ki | 4 | — | |
GFBKEXLXXAYEAN
|
6.5 | IC50 | 4 | — | |
RPXVIAFEQBNEAX
|
6.5 | IC50 | 4 | — | |
IAWXTSMHXFRLQR
|
6.5 | IC50 | 4 | — | |
OQCIHSFMLURANM
|
6.5 | IC50 | 5 | — | |
FTNICLJXPYLDAH
|
6.5 | IC50 | 3 | — | |
IYXKOVFPNWKUPM
|
6.5 | IC50 | 3 | — | |
PNHHRWFIFSETRC
|
6.5 | IC50 | 2 | — | |
XTASTURWHDUENT
|
6.4 | IC50 | 2 | — | |
FACUYWPMDKTVFU
|
6.4 | Ki | 2 | — | |
FNXUJFFLRGBKLM
|
6.4 | Ki | 4 | — | |
VUYXWDSZUHMHRT
|
6.4 | Ki | 4 | — | |
ZKAVBWHGBZBUAU
|
6.4 | IC50 | 2 | — | |
JLUIVZIFGHVQKL
|
6.4 | IC50 | 4 | — | |
BICPPLXRHOQXDM
|
6.3 | Ki | 4 | — | |
WHUUTDBJXJRKMK
|
6.3 | IC50 | 20 | — | |
YZSBXDRTJNDPDR
|
6.3 | IC50 | 4 | — | |
MDDDAYFWAQDGRP
|
6.3 | IC50 | 2 | — | |
VTWXNIYVJOMEKC
|
6.3 | Ki | 4 | — | |
DRSBUYJJPSUTFO
|
6.3 | Ki | 4 | — | |
XTTJVGFNQFHWPI
|
6.2 | IC50 | 4 | — | |
QBCVGLJGAYPHNK
|
6.2 | Ki | 4 | — | |
MQFAYNCEKGLLKI
|
6.2 | IC50 | 4 | — | |
WXUBLMKEFDTLAG
|
6.2 | Ki | 4 | — | |
NZJUQOAVHJUPHZ
|
6.2 | IC50 | 4 | — | |
AYWSXMRAQKWRMH
|
6.2 | Ki | 3 | — | |
GEEFQPZFVXQGCJ
|
6.2 | IC50 | 4 | — | |
GXLYWXMBTOIUTQ
|
6.2 | IC50 | 4 | — | |
KZFIZNJSPIBCFN
|
6.2 | Ki | 4 | — | |
ZPJJGAUEQIVPRW
|
6.2 | IC50 | 4 | — | |
LUIPVVRVNKNJEK
|
6.1 | Ki | 5 | — | |
YGSXLTANQIVRPQ
|
6.1 | IC50 | 4 | — | |
LBRZSCJIEHCPKW
|
6.1 | Ki | 4 | — | |
OOIMGNLMHOCHOG
|
6.1 | Ki | 4 | — | |
IFNJBSHPAUZGBB
|
6.0 | Ki | 4 | — | |
MCKOVZZCGOMMIB
|
6.0 | Ki | 6 | — | |
LPMRCCNDNGONCD
|
6.0 | IC50 | 11 | — | |
ROBLGUMDXHEHOO
|
6.0 | Ki | 4 | — | |
VIROLUKPVOVJDX
|
6.0 | Ki | 4 | — |