Target Details
| UniProt AC | P42229 |
|---|---|
| Gene Symbol | STAT5A |
| Protein Name | Signal transducer and activator of transcription 5A |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00017 (SH2) PF01017 (STAT_alpha) PF02864 (STAT_bind) PF02865 (STAT_int) PF21354 (STAT_linker) |
Summary
- Multi-target molecules 11
- Clinical molecules 2
- Avg pChEMBL 7.09
KEGG Pathways (18)
- AGE-RAGE signaling pathway in diabetic complications
- Acute myeloid leukemia
- Chemical carcinogenesis - receptor activation
- Chronic myeloid leukemia
- ErbB signaling pathway
- Growth hormone synthesis, secretion and action
- Hepatitis B
- Hormone signaling
- Human T-cell leukemia virus 1 infection
- JAK-STAT signaling pathway
- Measles
- Necroptosis
- Non-small cell lung cancer
- Pathways in cancer
- Prolactin signaling pathway
- Th1 and Th2 cell differentiation
- Th17 cell differentiation
- Viral carcinogenesis
Active Molecules (11)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
MWKSRKSEWLRPBL
|
8.4 | Kd | 1075 | — | |
SLCFEJAMCRLYRG
|
8.3 | IC50 | 8 | Yes | |
UIARLYUEJFELEN
|
8.0 | IC50 | 289 | Yes | |
PDOQBOJDRPLBQU
|
7.5 | IC50 | 21 | — | |
KIMCXIRMMLNCFO
|
7.4 | IC50 | 8 | — | |
NLGFHGWLXCBAQB
|
7.2 | IC50 | 8 | — | |
TXBCKCGOGPLPMZ
|
6.7 | IC50 | 8 | — | |
VFPYGNNOSJWBHF
|
6.3 | Kd | 2 | — | |
BZSUCLDZAQTFQJ
|
6.2 | IC50 | 4 | — | |
KJJHAYNANYPNEE
|
6.0 | Ki | 2 | — | |
QOYWPVULYMHMHY
|
6.0 | Ki | 2 | — |