Target Details
| UniProt AC | P41972 |
|---|---|
| Gene Symbol | ileS |
| Protein Name | Isoleucine--tRNA ligase |
| Organism | Staphylococcus aureus |
| Entry Name | |
| Organism Category | Pathogen |
| Pfam Domains | PF08264 (Anticodon_1) PF00133 (tRNA-synt_1) PF06827 (zf-FPG_IleRS) |
Summary
- Multi-target molecules 13
- Clinical molecules 0
- Avg pChEMBL 6.97
Active Molecules (13)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
HDXFGBFIEQUETL
|
7.8 | IC50 | 2 | — | |
XQLMQZYDYIYOIJ
|
7.4 | IC50 | 2 | — | |
QMWNPOPSMQKQAL
|
7.4 | IC50 | 2 | — | |
SKMGGGPZQRRMTG
|
7.3 | IC50 | 2 | — | |
FUNOATJOTYEZJZ
|
7.0 | IC50 | 2 | — | |
FREGHQKQLWGWHX
|
7.0 | IC50 | 2 | — | |
WNORCWSRNMBRBU
|
7.0 | IC50 | 2 | — | |
WAXQESJXPPKIIV
|
6.9 | IC50 | 2 | — | |
WCVCPXUETPTILF
|
6.9 | IC50 | 2 | — | |
ORNSGNNIYULCMK
|
6.6 | IC50 | 2 | — | |
VMXXHKARGFATOU
|
6.6 | IC50 | 2 | — | |
XSRXZXOKBZFCHB
|
6.5 | IC50 | 2 | — | |
YABWOCJHKKFQIN
|
6.0 | IC50 | 3 | — |