Target Details
UniProt ACP41968
Gene SymbolMC3R
Protein NameMelanocortin receptor 3
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 557
  • Clinical molecules 0
  • Avg pChEMBL 7.19
Associated Diseases (1)
Top Co-occurrence Targets
Active Molecules (557)
InChIKey pChEMBL Type Targets Clinical
RNCVEEUMKRRHLC 8.5 IC50 4
UKMQKNTZNHDSPD 8.5 IC50 4
KIFNALNSUOJQPJ 8.5 Ki 4
AETQUGIIFBPWMW 8.5 Ki 2
BBJOQSQVKOIBHK 8.5 IC50 4
RDCIPOBDQMOUKD 8.5 IC50 4
ZRHYLFBORVIBEU 8.5 Ki 3
GGYWLZFXFKFWKL 8.4 IC50 4
VGBVAARMQYYITG 8.4 Ki 3
YLVUKTHOPXMSDE 8.4 Ki 2
ONUUGLJKQIIBGJ 8.4 IC50 3
KHGZKFBKKYRZCD 8.4 IC50 3
RVEIEULWMVBMRD 8.4 IC50 4
ZRCSDDHAGXRMLM 8.4 IC50 4
GGYWLZFXFKFWKL 8.3 IC50 3
NVIBFTUPAARCBA 8.3 Kd 2
OKHXBJLIBJDJMV 8.3 IC50 4
QXRXXIKAVZAGHZ 8.3 IC50 3
WSDYWWDQJYPQDS 8.3 IC50 4
YXIBEMYOGWJEQC 8.3 Ki 4
ZWTUZOQCWSYYNO 8.3 IC50 3
KLOVFBFHFHKKJQ 8.3 IC50 3
MZFOEDJULWOZIV 8.3 IC50 3
AMLJFTMENZUCBN 8.3 Ki 3
DPJAKAHREXIEPH 8.2 IC50 3
JKPIUTPQBDXSRH 8.2 Ki 3
FHNLUGMXKXPEFR 8.2 IC50 4
OHFMRHZLQMSCRN 8.2 IC50 4
TYFFXNLNRYRUAU 8.2 IC50 3
SOCBNUUFEBTEOP 8.2 IC50 3
GZWUQPQBOGLSIM 8.2 IC50 3
KLOVFBFHFHKKJQ 8.2 IC50 3
UKCAJRRGLXHDRO 8.2 Ki 3
UVUOMESIOOEXGA 8.2 IC50 3
LZYYGZAXFMYSBE 8.2 Ki 4
SLEIICTWQFRIFM 8.2 Ki 3
YZQBDVJPOXNSJR 8.2 Ki 3
SQKAQIVUMGJDFA 8.1 Ki 2
BINHUIMAVHQSOM 8.1 Ki 4
MTFOEQYGYVFQPJ 8.1 Ki 3
NEVVXMYOTHZJES 8.1 IC50 3
PPKIGEMCDOLKEY 8.1 Ki 3
PPKIGEMCDOLKEY 8.1 Ki 3
YENCSZMEVJAKQJ 8.1 IC50 4
SNEMRJZDOOLWPZ 8.1 Ki 4
GGYWLZFXFKFWKL 8.1 IC50 3
HOWXKXAJVJPQOI 8.1 IC50 3
SLPDXDVCXNVEEV 8.1 Ki 2
HDBFFTYMERRCIX 8.0 IC50 3
XQMPAWYRHAOJTE 8.0 Ki 4
2D structure