Target Details
| UniProt AC | P41968 |
|---|---|
| Gene Symbol | MC3R |
| Protein Name | Melanocortin receptor 3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00001 (7tm_1) |
Summary
- Multi-target molecules 557
- Clinical molecules 0
- Avg pChEMBL 7.19
KEGG Pathways (3)
Associated Diseases (1)
Active Molecules (557)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
XDLJELQQEILLFZ
|
10.0 | Ki | 4 | — | |
JNEKRCCXHUFBPL
|
9.7 | IC50 | 3 | — | |
QXDWLOZJHHTTCF
|
9.7 | IC50 | 3 | — | |
KRZXMSMNMZEKGP
|
9.7 | Ki | 4 | — | |
BUVGQEXSQXRZQG
|
9.6 | Ki | 4 | — | |
GGYWLZFXFKFWKL
|
9.6 | Ki | 3 | — | |
QXDWLOZJHHTTCF
|
9.5 | IC50 | 3 | — | |
YIYFGSBFHVAQLI
|
9.4 | Ki | 2 | — | |
JNEKRCCXHUFBPL
|
9.4 | IC50 | 3 | — | |
RANDNDRFMFBRFD
|
9.2 | Ki | 3 | — | |
JMFDAPXKXHNPIL
|
9.0 | Ki | 3 | — | |
FJSKRKLUQFIKJP
|
9.0 | Ki | 3 | — | |
KYOVLZCJSUXUJI
|
9.0 | Ki | 3 | — | |
UMHVNRYGRKBTCG
|
9.0 | IC50 | 4 | — | |
ZSAXEKUGMLDFHT
|
9.0 | Ki | 3 | — | |
AXYNQPYLILCAPC
|
9.0 | Ki | 3 | — | |
CBZNNNCTDMTAGU
|
9.0 | Ki | 3 | — | |
ILTSJNSAHXKVSQ
|
8.9 | Ki | 3 | — | |
KPKOJXZVOJTTBP
|
8.9 | IC50 | 2 | — | |
ODSFZEXVNOIJHI
|
8.9 | IC50 | 3 | — | |
UAHFGYDRQSXQEB
|
8.9 | IC50 | 5 | — | |
ZPANOUCVWZTSLE
|
8.9 | IC50 | 4 | — | |
LBOGVWLKUREGLH
|
8.9 | IC50 | 2 | — | |
TUOOEJAUOYDGGA
|
8.8 | IC50 | 4 | — | |
ZSONGANRJTVTCP
|
8.8 | Ki | 4 | — | |
ZTSQVRSYAGAZPG
|
8.8 | IC50 | 4 | — | |
AKHYEKNKKQDKLB
|
8.8 | IC50 | 2 | — | |
DLVAKQPHOINITK
|
8.8 | IC50 | 4 | — | |
UCOANIAEMBZDQE
|
8.8 | IC50 | 2 | — | |
GVZTZLFKKLVBJF
|
8.8 | IC50 | 3 | — | |
JDKLPDJLXHXHNV
|
8.7 | IC50 | 4 | — | |
KWBYYFKCXHSTPA
|
8.7 | IC50 | 4 | — | |
QBYHLGIJWBFDGJ
|
8.7 | IC50 | 4 | — | |
RVKSMTBVJXMWFD
|
8.7 | IC50 | 4 | — | |
UBKGFMZTCLCOLM
|
8.7 | Ki | 4 | — | |
REMHNXQVRVXAGT
|
8.7 | IC50 | 4 | — | |
RQCWCCUAQKMWGM
|
8.7 | IC50 | 4 | — | |
GGYWLZFXFKFWKL
|
8.6 | IC50 | 4 | — | |
REMHNXQVRVXAGT
|
8.6 | IC50 | 4 | — | |
GJFLVESIDOAAJH
|
8.6 | IC50 | 2 | — | |
OMSSRUBSGSKAFS
|
8.6 | IC50 | 3 | — | |
KHGZKFBKKYRZCD
|
8.6 | IC50 | 3 | — | |
NEVVXMYOTHZJES
|
8.6 | IC50 | 3 | — | |
XMQSVPKHHVWBGS
|
8.6 | IC50 | 4 | — | |
XTFWFFODDNNYFQ
|
8.6 | Ki | 4 | — | |
UHCXNXMBPAFWDS
|
8.6 | IC50 | 3 | — | |
XUCSIJVANOTEDW
|
8.6 | Ki | 3 | — | |
UMHVNRYGRKBTCG
|
8.6 | IC50 | 4 | — | |
GYFGNZUSQUDKII
|
8.5 | IC50 | 3 | — | |
NVIBFTUPAARCBA
|
8.5 | IC50 | 3 | — |