Target Details
UniProt ACP41743
Gene SymbolPRKCI
Protein NameProtein kinase C iota type
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00130 (C1_1) PF00564 (PB1) PF00069 (Pkinase) PF00433 (Pkinase_C)
Summary
  • Multi-target molecules 158
  • Clinical molecules 94
  • Avg pChEMBL 7.1
Top Co-occurrence Targets
Active Molecules (158)
InChIKey pChEMBL Type Targets Clinical
LWSORTKUYSYDMP 6.0 IC50 12
MAHFVAHPQSLLJF 6.0 IC50 288
MASJMHFQMYAPJR 6.0 Ki 41
MHHTXOIOMYDUOQ 6.0 Ki 4
NJPWCTYVEJIQBM 6.0 Ki 72
NKANXQFJJICGDU 6.0 IC50 35 Yes
RQVKVJIRFKVPBF 6.0 Ki 13
UUCJUCRTIKZRFG 6.0 IC50 12 Yes
2D structure