Target Details
| UniProt AC | P41743 |
|---|---|
| Gene Symbol | PRKCI |
| Protein Name | Protein kinase C iota type |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00130 (C1_1) PF00564 (PB1) PF00069 (Pkinase) PF00433 (Pkinase_C) |
Summary
- Multi-target molecules 158
- Clinical molecules 94
- Avg pChEMBL 7.1
KEGG Pathways (8)
Active Molecules (158)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
KOZFSFOOLUUIGY
|
6.6 | IC50 | 26 | — | |
QMGUOJYZJKLOLH
|
6.6 | IC50 | 21 | Yes | |
SSZFVGXDYBMVDD
|
6.6 | IC50 | 12 | Yes | |
UMTWTCVTRDYHQQ
|
6.6 | Ki | 56 | — | |
NXSJMRCTGYTSTK
|
6.6 | Kd | 200 | — | |
PBCZSGKMGDDXIJ
|
6.6 | IC50 | 12 | Yes | |
LAOIBIIMKUINJL
|
6.6 | IC50 | 12 | Yes | |
IXOVKVHWGKDXKQ
|
6.6 | IC50 | 12 | Yes | |
BRZYOTMFHLERHD
|
6.5 | Ki | 17 | Yes | |
XNKIVXYFRPYKHO
|
6.5 | IC50 | 12 | Yes | |
OSVUGUHRKMMBSE
|
6.5 | Kd | 170 | — | |
TVIALAOHRQNPOI
|
6.5 | IC50 | 12 | Yes | |
HPCPUHOULFPBCQ
|
6.5 | IC50 | 12 | Yes | |
JDZXLEPJWLCESI
|
6.5 | IC50 | 12 | Yes | |
RHBWAFDCVFMIFK
|
6.5 | IC50 | 12 | Yes | |
HKSZLNNOFSGOKW
|
6.4 | IC50 | 49 | Yes | |
RPLXVENRWORMRX
|
6.4 | IC50 | 12 | Yes | |
BMGQWWVMWDBQGC
|
6.4 | IC50 | 147 | Yes | |
MQFYZWYYZGTHAN
|
6.4 | IC50 | 14 | — | |
OAVGBZOFDPFGPJ
|
6.4 | Ki | 42 | Yes | |
OUJZYQBEFNDJQN
|
6.4 | Ki | 71 | — | |
KAJXOWFGKYKMMZ
|
6.4 | IC50 | 26 | Yes | |
ZFNQOYBHHLGQDV
|
6.3 | IC50 | 12 | Yes | |
BMBIKZHGTPMMMM
|
6.3 | IC50 | 14 | — | |
CPRVBHBRBVVLHL
|
6.3 | IC50 | 11 | — | |
ATBAETXFFCOZOY
|
6.3 | IC50 | 39 | — | |
CCRCRSXDKXZDGK
|
6.3 | IC50 | 12 | Yes | |
XYZNKCSDQRKAFR
|
6.3 | Ki | 53 | — | |
JSPAUBUYPPZXSG
|
6.3 | Ki | 17 | Yes | |
ORNADCNXUPZOQN
|
6.3 | IC50 | 15 | — | |
NEGCBIBMPAHBIM
|
6.3 | IC50 | 12 | Yes | |
BAQFZMFDZMQJAM
|
6.2 | IC50 | 12 | Yes | |
IQTLSOGTQGJADC
|
6.2 | IC50 | 2 | — | |
TXBFOGDMTCNBBT
|
6.2 | IC50 | 12 | Yes | |
HLXIFVDYTGEUJV
|
6.2 | IC50 | 15 | Yes | |
KPJDEGAKXAUVAC
|
6.2 | Ki | 15 | Yes | |
CWFIQHQECWPWQG
|
6.2 | IC50 | 16 | Yes | |
ORNADCNXUPZOQN
|
6.2 | IC50 | 15 | — | |
NGFGTMFVWSDFPS
|
6.1 | IC50 | 32 | — | |
AXTAPYRUEKNRBA
|
6.1 | IC50 | 24 | — | |
RKUKAACYUCUJEE
|
6.1 | Ki | 58 | — | |
WSXYBDKZFNJOTP
|
6.1 | IC50 | 12 | Yes | |
MRBNLCLXWRXFJX
|
6.1 | IC50 | 15 | — | |
GHRBXKFGXPOEGA
|
6.0 | IC50 | 12 | Yes | |
KUYKGKWALOSLME
|
6.0 | IC50 | 2 | — | |
YAZWNGDLKIJVLM
|
6.0 | IC50 | 2 | — | |
CHTMRWQLNNRRFJ
|
6.0 | Ki | 70 | — | |
HSKVRPZJBMXFDX
|
6.0 | Ki | 20 | — | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — | |
KHVVJKLNKLQLJZ
|
6.0 | IC50 | 288 | — |