Target Details
| UniProt AC | P41743 |
|---|---|
| Gene Symbol | PRKCI |
| Protein Name | Protein kinase C iota type |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00130 (C1_1) PF00564 (PB1) PF00069 (Pkinase) PF00433 (Pkinase_C) |
Summary
- Multi-target molecules 158
- Clinical molecules 94
- Avg pChEMBL 7.1
KEGG Pathways (8)
Active Molecules (158)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
NTUVEMUMVHHACY
|
7.4 | IC50 | 12 | Yes | |
KOZFSFOOLUUIGY
|
7.3 | IC50 | 88 | Yes | |
WKZTVBCDQYBGBO
|
7.3 | IC50 | 16 | Yes | |
RFUHKEPWGZUNBG
|
7.3 | IC50 | 4 | — | |
BMGQWWVMWDBQGC
|
7.3 | IC50 | 91 | Yes | |
MDHNNGDJYHAYKJ
|
7.3 | IC50 | 12 | Yes | |
XXIWRTOLXWAEJC
|
7.2 | IC50 | 13 | Yes | |
IJNGXROUMFEKDB
|
7.2 | Ki | 39 | — | |
TUBBFDZWFNUZLH
|
7.2 | IC50 | 12 | Yes | |
NRUVICOXXLOXCB
|
7.2 | IC50 | 13 | Yes | |
VKQMYKOSLRYFTF
|
7.2 | IC50 | 2 | — | |
MGMNDPRNDCWSMZ
|
7.2 | IC50 | 12 | Yes | |
TXGUECVFNFKTBD
|
7.2 | IC50 | 2 | — | |
GRENHRYHWHSBLM
|
7.1 | IC50 | 12 | Yes | |
LGCKGDRUTNACTA
|
7.1 | IC50 | 11 | — | |
OFPFIAWWDTYSBZ
|
7.1 | Ki | 15 | Yes | |
RHLRPKGACJKWPF
|
7.1 | IC50 | 12 | Yes | |
GGQAEINRBKFRGZ
|
7.1 | IC50 | 15 | Yes | |
NHDDTLMPCVOXFH
|
7.1 | IC50 | 16 | Yes | |
SXDPQGRNHSLZPC
|
7.0 | IC50 | 18 | — | |
MQCCJEYZKWZQHU
|
7.0 | IC50 | 15 | Yes | |
YSVVBGPTTSJYPA
|
7.0 | IC50 | 13 | Yes | |
PFAZIMNYEBJHOA
|
7.0 | IC50 | 12 | Yes | |
VVENTSJOKWJQFG
|
7.0 | IC50 | 2 | — | |
XRFOMFNAMTYCFF
|
7.0 | IC50 | 12 | Yes | |
YUAWUNMKPARPJD
|
7.0 | IC50 | 14 | Yes | |
LASNFRKYDHLWNQ
|
7.0 | IC50 | 3 | — | |
KOZFSFOOLUUIGY
|
6.9 | IC50 | 15 | Yes | |
OGJTZCZJWZSZBT
|
6.9 | IC50 | 12 | Yes | |
VWHZWDRIMLETBG
|
6.9 | IC50 | 12 | Yes | |
DRCBMJUPXHWGMN
|
6.8 | IC50 | 15 | Yes | |
QNULKTUETCUJKC
|
6.8 | IC50 | 14 | Yes | |
CZIVUSJISIAXJB
|
6.8 | IC50 | 18 | — | |
OOPMDKIRVTXOPT
|
6.8 | IC50 | 11 | — | |
JCHWETQOLSPUBV
|
6.8 | IC50 | 14 | — | |
JHKZENPNLYAVCT
|
6.8 | IC50 | 15 | Yes | |
VWVYILCFSYNJHF
|
6.8 | IC50 | 49 | — | |
ZCCPLJOKGAACRT
|
6.8 | Kd | 599 | — | |
OQSTWXKHTZWKLD
|
6.8 | IC50 | 15 | Yes | |
DQYBRTASHMYDJG
|
6.7 | IC50 | 13 | Yes | |
LGSHHKIOBFPSEK
|
6.7 | IC50 | 12 | Yes | |
XPHWIERLJBFPFV
|
6.7 | Ki | 69 | — | |
NTXWXFSAJRMWNA
|
6.7 | IC50 | 15 | — | |
RAOJISQDGOOXTK
|
6.7 | IC50 | 14 | Yes | |
MEXUTNIFSHFQRG
|
6.7 | IC50 | 21 | Yes | |
GZJKVFKNTQXSQM
|
6.7 | IC50 | 12 | Yes | |
MZNUNTIEUOYNNT
|
6.6 | IC50 | 12 | Yes | |
OXEOHAXVZADDOC
|
6.6 | IC50 | 12 | Yes | |
YSVVBGPTTSJYPA
|
6.6 | IC50 | 12 | Yes | |
KGPGFQWBCSZGEL
|
6.6 | Kd | 59 | Yes |