Target Details
| UniProt AC | P41597 |
|---|---|
| Gene Symbol | CCR2 |
| Protein Name | C-C chemokine receptor type 2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00001 (7tm_1) |
Summary
- Multi-target molecules 187
- Clinical molecules 0
- Avg pChEMBL 7.65
KEGG Pathways (3)
Associated Diseases (2)
Active Molecules (187)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
UVLRQIJLSWXUPM
|
6.8 | Ki | 2 | — | |
LFEZDWBBQLHEMC
|
6.8 | IC50 | 2 | — | |
TWDSSLGDUOHXCF
|
6.8 | IC50 | 3 | — | |
COCOWIOUVHRNJM
|
6.8 | Ki | 2 | — | |
UWKZCWZZZAHBSF
|
6.8 | Ki | 2 | — | |
VKUIPZIEQFUJHB
|
6.8 | Ki | 2 | — | |
XJDNAMFCUOWNRL
|
6.8 | IC50 | 2 | — | |
BKQDNXBGUIWZEK
|
6.8 | Ki | 2 | — | |
DTYWPXSMHVEQQW
|
6.7 | IC50 | 2 | — | |
YLNOGPJREAMGJN
|
6.7 | IC50 | 2 | — | |
RMFBDGDNDXDJJH
|
6.7 | Ki | 2 | — | |
DNMIVGPRKRLQLY
|
6.7 | Ki | 2 | — | |
GCFPGFUOEIYTMZ
|
6.7 | Ki | 2 | — | |
VDMUUPCXLAKUJY
|
6.7 | Ki | 2 | — | |
AYEWGKWGWGVEHB
|
6.6 | Ki | 2 | — | |
MEKUTHVEROQRGI
|
6.6 | Ki | 2 | — | |
PUKIAWNJPGVZPZ
|
6.5 | Ki | 2 | — | |
IKYXYVLOGJLJTF
|
6.4 | Ki | 2 | — | |
XOXUVAJFNVIHLG
|
6.4 | Ki | 2 | — | |
DNPRHSLKGYTIJX
|
6.3 | IC50 | 2 | — | |
VZPTWPGJCWIVGK
|
6.3 | Ki | 2 | — | |
SWGQDPWKPYZEEH
|
6.1 | IC50 | 2 | — | |
IWSNTIDXIKYXSU
|
6.1 | Ki | 2 | — | |
HYIMSNHJOBLJNT
|
6.1 | Ki | 6 | — | |
AFZSMODLJJCVPP
|
6.0 | Ki | 12 | — | |
BOHSWBWGIHBCLE
|
6.0 | IC50 | 2 | — | |
AUZONCFQVSMFAP
|
6.0 | Ki | 15 | — | |
JLWTUPLIJAHTKE
|
6.0 | IC50 | 3 | — | |
JQCWNEXLKSGUJQ
|
6.0 | IC50 | 3 | — | |
KDILGLNJDNVPLP
|
6.0 | IC50 | 3 | — | |
KRZMKLFPGBUXGH
|
6.0 | IC50 | 3 | — | |
MBEYXNMHPBPYSU
|
6.0 | IC50 | 3 | — | |
NVDYRDZHCINQQB
|
6.0 | IC50 | 3 | — | |
PUDPIQFNZNNYGT
|
6.0 | IC50 | 3 | — | |
QANOXOWLUOTIAC
|
6.0 | IC50 | 3 | — | |
UCJIXVPTONWDEH
|
6.0 | IC50 | 3 | — | |
VYZJFSWYQODVMI
|
6.0 | IC50 | 3 | — |