Target Details
| UniProt AC | P41597 |
|---|---|
| Gene Symbol | CCR2 |
| Protein Name | C-C chemokine receptor type 2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00001 (7tm_1) |
Summary
- Multi-target molecules 187
- Clinical molecules 0
- Avg pChEMBL 7.65
KEGG Pathways (3)
Associated Diseases (2)
Active Molecules (187)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
YIQPUIGJQJDJOS
|
10.2 | IC50 | 5 | — | |
MTBTXJDOIZCIGH
|
9.4 | IC50 | 2 | — | |
PJTGSIKANITYOO
|
9.4 | IC50 | 2 | — | |
WKTVEPAXEKXDKZ
|
9.4 | Ki | 2 | — | |
BXZCHELXYNXCDS
|
9.3 | Ki | 2 | — | |
ZILPZMJIIYWEIE
|
9.3 | IC50 | 2 | — | |
MTMDXAIUENDNDL
|
9.3 | Kd | 2 | — | |
DECZUBPHXAXNSH
|
9.2 | Ki | 2 | — | |
FVNQVTADUDKSGZ
|
9.2 | Ki | 2 | — | |
SNVMTABEFLKIEG
|
9.2 | IC50 | 2 | — | |
GVOISEJVFFIGQE
|
9.2 | IC50 | 2 | — | |
NUJWKQSEJDYCDB
|
9.2 | IC50 | 4 | — | |
NIGNHDUWKZDZLS
|
9.1 | IC50 | 2 | — | |
BYVKUTDQYZLLAZ
|
9.1 | IC50 | 2 | — | |
CJGHKRWUTQLMOP
|
9.1 | IC50 | 2 | — | |
CSTRIVMEIYPLGJ
|
9.0 | Ki | 2 | — | |
FFBYNQCXDQNNQT
|
9.0 | Ki | 2 | — | |
OKIJQELRSBSEJX
|
9.0 | IC50 | 2 | — | |
GQLXQNMFKWOOSD
|
8.9 | Ki | 3 | — | |
JEUSLIAZMCQUCV
|
8.9 | IC50 | 2 | — | |
UAKDPJAUOVRMIX
|
8.9 | IC50 | 2 | — | |
QAPTWHXHEYAIKG
|
8.8 | IC50 | 2 | — | |
KLBHHUODQVCBKX
|
8.8 | Ki | 2 | — | |
SSYDLAOTEQIPAM
|
8.8 | Ki | 2 | — | |
CHNSDJOKVUZBQF
|
8.7 | Ki | 2 | — | |
HKIFMAJLMSGIOP
|
8.7 | Ki | 2 | — | |
QOYZHUQEWFRBJB
|
8.7 | IC50 | 2 | — | |
AQTIPNCIMOFYSH
|
8.7 | IC50 | 2 | — | |
SCSTUPQPTWXCHZ
|
8.7 | Ki | 2 | — | |
COTMDVGGTIZRGD
|
8.6 | Ki | 2 | — | |
DEXJQUDODNDJEZ
|
8.6 | IC50 | 2 | — | |
LAPGFBUSBADRJT
|
8.6 | IC50 | 2 | — | |
BCRSYZQXPRWUJQ
|
8.6 | IC50 | 3 | — | |
HTGCOGKGWKXISK
|
8.6 | IC50 | 2 | — | |
NMYCPGLFRHGTSV
|
8.6 | IC50 | 2 | — | |
QJQMEUAVQLMKRZ
|
8.5 | IC50 | 2 | — | |
YEQFSCLZXBNXBX
|
8.5 | IC50 | 2 | — | |
OIGUMNDUYFBXEM
|
8.5 | Ki | 3 | — | |
DNPRHSLKGYTIJX
|
8.5 | IC50 | 2 | — | |
DQWSENNLMPJNRJ
|
8.5 | IC50 | 2 | — | |
WXRJQYAAIDCOMB
|
8.5 | IC50 | 2 | — | |
YIQYJBKGDDWABP
|
8.5 | IC50 | 2 | — | |
YLVBQGLIQXQGPH
|
8.4 | IC50 | 2 | — | |
NABAWBCHPQOSTO
|
8.4 | Ki | 2 | — | |
ILPQLCKGOBBIPI
|
8.4 | IC50 | 2 | — | |
OOGWCCRYNCAIBK
|
8.4 | IC50 | 2 | — | |
MZEOSVPWMSEFPW
|
8.4 | IC50 | 2 | — | |
CMVHFGNTABZQJU
|
8.3 | IC50 | 2 | — | |
PNDKCRDVVKJPKG
|
8.2 | IC50 | 2 | — | |
PNDKCRDVVKJPKG
|
8.2 | IC50 | 3 | — |