Target Details
| UniProt AC | P41586 |
|---|---|
| Gene Symbol | ADCYAP1R1 |
| Protein Name | Pituitary adenylate cyclase-activating polypeptide type I receptor |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00002 (7tm_2) PF02793 (HRM) |
Summary
- Multi-target molecules 12
- Clinical molecules 0
- Avg pChEMBL 7.74
KEGG Pathways (5)
Active Molecules (12)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
UFTCZKMBJOPXDM
|
9.0 | IC50 | 2 | — | |
GDQXRMJXFNQXMJ
|
8.5 | IC50 | 3 | — | |
HXROOIDQCQSPGK
|
8.5 | IC50 | 3 | — | |
HVFBYLQDWMQSMM
|
8.3 | IC50 | 3 | — | |
RZGBUJXSKLDAFE
|
8.2 | IC50 | 3 | — | |
IAWMQYIXAKXMGI
|
8.0 | IC50 | 2 | — | |
UFKWYYSODZYURD
|
7.3 | IC50 | 3 | — | |
AFKHWKJSOKSDOT
|
7.2 | IC50 | 2 | — | |
ZGRAABYQGYPWLS
|
7.2 | Ki | 2 | — | |
PKTPZIVUKIRQDY
|
7.2 | IC50 | 3 | — | |
HNTXQDRFWJBZGO
|
7.1 | Ki | 2 | — | |
JJGVEWLQTOEULJ
|
6.2 | Ki | 2 | — |