Target Details
| UniProt AC | P41279 |
|---|---|
| Gene Symbol | MAP3K8 |
| Protein Name | Mitogen-activated protein kinase kinase kinase 8 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 15
- Clinical molecules 2
- Avg pChEMBL 7.32
KEGG Pathways (4)
Active Molecules (15)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
PHNZIIMWDVXPGG
|
8.8 | IC50 | 2 | — | |
PXRDIWAVNLQFBI
|
8.7 | IC50 | 6 | Yes | |
HIASHEATKNRFJC
|
8.2 | IC50 | 2 | Yes | |
KEZDJRADZYWSSG
|
7.7 | IC50 | 2 | — | |
HFOOHVUKODGHBP
|
7.7 | IC50 | 2 | — | |
GRPUCYCKBBWGEO
|
7.7 | IC50 | 2 | — | |
FYBDFTOKGKWXLM
|
7.6 | IC50 | 2 | — | |
IKMGVUYZBWHRNX
|
7.4 | IC50 | 2 | — | |
NMEUKWOOQOHUNA
|
7.3 | IC50 | 6 | — | |
NCPSMBVBKJXJPP
|
6.9 | IC50 | 3 | — | |
NHXNHCQTGVIMIV
|
6.7 | IC50 | 2 | — | |
YUYWSKXPXLUJNA
|
6.4 | IC50 | 2 | — | |
PQVDKUZOKMCUSV
|
6.4 | IC50 | 3 | — | |
ULMZCAWRPCELOE
|
6.2 | IC50 | 3 | — | |
IWDISKBCTNXZQH
|
6.0 | IC50 | 3 | — |