Target Details
| UniProt AC | P41240 |
|---|---|
| Gene Symbol | CSK |
| Protein Name | Tyrosine-protein kinase CSK |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07714 (PK_Tyr_Ser-Thr) PF00017 (SH2) PF00018 (SH3_1) |
Summary
- Multi-target molecules 104
- Clinical molecules 13
- Avg pChEMBL 7.23
KEGG Pathways (2)
Active Molecules (104)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — | |
KHVVJKLNKLQLJZ
|
6.0 | IC50 | 288 | — | |
MAHFVAHPQSLLJF
|
6.0 | IC50 | 288 | — | |
MWKSRKSEWLRPBL
|
6.0 | Kd | 1075 | — |