Target Details
UniProt ACP41240
Gene SymbolCSK
Protein NameTyrosine-protein kinase CSK
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF07714 (PK_Tyr_Ser-Thr) PF00017 (SH2) PF00018 (SH3_1)
Summary
  • Multi-target molecules 104
  • Clinical molecules 13
  • Avg pChEMBL 7.23
Top Co-occurrence Targets
Active Molecules (104)
InChIKey pChEMBL Type Targets Clinical
ZBNZXTGUTAYRHI 9.0 Kd 102 Yes
SYWUIAOLWMUYTP 8.8 IC50 3
DEGODTVDGRTRCG 8.7 IC50 2
LCYSSHSIKSARGO 8.7 IC50 19
XYFPWWZEPKGCCK 8.6 IC50 34
SSDFTYWIYVWCIE 8.6 IC50 17
YQDGGVYOYHQDIX 8.5 IC50 2
LQQYARMJQBHKQQ 8.4 IC50 2
NQWJYXLLLYRYCZ 8.4 IC50 2
ZLXUXNOXPKFKQF 8.4 IC50 2
HNWZKSBXLQWJOE 8.3 IC50 3
OROLCINTIPDVAI 8.3 IC50 2
QRHLGEHZPDSLFJ 8.3 IC50 2
CMJGHWQDYMQXML 8.2 IC50 2
KMKHVCGUHDWGJX 8.2 IC50 2
RWCFKPKDVWBGSU 8.2 IC50 2
KSUDUUBCXJUFRL 8.2 Kd 12
RPQORVRVHTUMJD 8.1 IC50 2
UCOFLDBJVAAAFU 8.1 IC50 2
PUKGRYCUACBXDB 8.1 IC50 2
YHVHYWYQEFELOW 8.1 IC50 44
LNVFYQLXYPFVNQ 8.0 IC50 2
FQCRNGFAAPZXFR 7.9 IC50 2
FYLYZGYKYWJXEB 7.9 IC50 2
PPCIDOUXWYIBPO 7.9 IC50 6
PHXJVRSECIGDHY 7.9 IC50 59
LUCKLKMOCDVQCV 7.9 IC50 2
VZXKLZIEIOUSHQ 7.9 IC50 2
JDCXTBTYAGHEQT 7.8 IC50 2
BNRJMXPCHXXMHT 7.8 IC50 2
KMMUTXPSVYLUNZ 7.8 IC50 3
DPSNOZFUMXEANO 7.8 Kd 7
TYSQKGWYQQCUCN 7.7 IC50 2
UVELXPTUBUVDHL 7.7 IC50 2
LXWXQRLCBZDGSZ 7.6 IC50 2
CYCZSOQHBKKPCR 7.6 IC50 2
OWHLXTINLAVFEZ 7.6 IC50 2
QZTCIPMCYKMSIT 7.6 IC50 2
VYDPOZRBQLVESU 7.6 IC50 2
DAILMCHHPABCQU 7.6 IC50 2
JHDISIQMSVRVDG 7.5 IC50 2
SFCBIFOAGRZJNX 7.5 Kd 22
TUUBKLDDTMKOCQ 7.5 IC50 2
IOJROWSVDGSWME 7.5 IC50 2
OOMBFNDWQIGHEK 7.5 Kd 22
UDXNFTYLGDGKTL 7.5 IC50 2
OJEIECWWENNREZ 7.4 IC50 2
UYAIFLOXHBEIGZ 7.4 IC50 2
FDVSOQRNTAPCHB 7.4 IC50 7 Yes
LTWKJBFCYCDGCV 7.4 IC50 2
2D structure