Target Details
| UniProt AC | P41229 |
|---|---|
| Gene Symbol | KDM5C |
| Protein Name | Lysine-specific demethylase 5C |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF01388 (ARID) PF02373 (JmjC) PF02375 (JmjN) PF21323 (KDM5_C-hel) PF00628 (PHD) PF08429 (PLU-1) PF02928 (zf-C5HC2) |
Summary
- Multi-target molecules 108
- Clinical molecules 0
- Avg pChEMBL 6.96
Associated Diseases (1)
Active Molecules (108)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
VCITXXCATLNLDE
|
7.1 | IC50 | 4 | — | |
FJLXFYHDLHZPQK
|
7.0 | IC50 | 4 | — | |
OFBASLHLTNSWOV
|
7.0 | IC50 | 4 | — | |
ZNWWSWJQMFNZDV
|
7.0 | IC50 | 5 | — | |
QOMJHYUHYMCFHT
|
7.0 | IC50 | 4 | — | |
JKWOFYNSPFBQLX
|
7.0 | IC50 | 4 | — | |
QDNXWZJEOBANTA
|
6.9 | IC50 | 4 | — | |
AVFIHINZEZRGBL
|
6.9 | IC50 | 4 | — | |
VHUXANZSWRXPQK
|
6.9 | IC50 | 4 | — | |
ARDXICZNEUJDDE
|
6.9 | IC50 | 5 | — | |
BUTZNIHTVCLMKG
|
6.9 | IC50 | 4 | — | |
IDVBVEOFBRZZEI
|
6.9 | IC50 | 5 | — | |
PLQDLMAFBDRQSK
|
6.9 | IC50 | 4 | — | |
DSGOLESVOJUGOK
|
6.9 | IC50 | 4 | — | |
XYBBSEAKIBCXQV
|
6.9 | IC50 | 4 | — | |
FGIPAHGTFZFKQH
|
6.9 | IC50 | 4 | — | |
VIUFHKFDQXQPJV
|
6.8 | IC50 | 4 | — | |
YGOIGEVVZIZMBG
|
6.8 | IC50 | 3 | — | |
RRZDZCQQAMZZMU
|
6.8 | IC50 | 4 | — | |
WDLBUONJQGHSKT
|
6.8 | IC50 | 3 | — | |
NPAMRWDIMURYSE
|
6.8 | IC50 | 3 | — | |
QVELLOOBNULIGQ
|
6.7 | IC50 | 3 | — | |
WUBIIGDBLTUSQG
|
6.7 | IC50 | 5 | — | |
FQYVJQRHNLIPIK
|
6.7 | IC50 | 4 | — | |
JGRPKOGHYBAVMW
|
6.7 | IC50 | 13 | — | |
OZMKCTFOIBLWOO
|
6.7 | IC50 | 5 | — | |
WXFDDWMINUVYFL
|
6.7 | IC50 | 4 | — | |
FSICLPHOMOJFQK
|
6.7 | IC50 | 4 | — | |
YAWHCFISAFZXHF
|
6.7 | IC50 | 4 | — | |
JRDMCDIQZVMPPB
|
6.6 | IC50 | 4 | — | |
NEJVXTLMGJPXNG
|
6.6 | IC50 | 2 | — | |
OTYMAMBJVVRSCZ
|
6.5 | IC50 | 4 | — | |
JEHSMTZNFSEDBY
|
6.5 | IC50 | 2 | — | |
SSZGYIZGRDDQEH
|
6.5 | IC50 | 3 | — | |
XMPNGNYDXRKBIH
|
6.5 | IC50 | 2 | — | |
WNSMPEBHTSITSG
|
6.5 | IC50 | 3 | — | |
JJUBVVYZQHPFMF
|
6.4 | IC50 | 3 | — | |
OXELDRCVUWWSFZ
|
6.4 | IC50 | 3 | — | |
YIEUEKVBIVGYSC
|
6.4 | IC50 | 2 | — | |
WMPDPRRYFWPZOM
|
6.3 | IC50 | 4 | — | |
XRMBRQWBOICYRP
|
6.3 | IC50 | 4 | — | |
MJIVRKPEXXHNJT
|
6.3 | IC50 | 9 | — | |
AVZCPICCWKMZDT
|
6.3 | IC50 | 5 | — | |
JMAUMLMBIAXZPR
|
6.3 | IC50 | 4 | — | |
WXDMSMYTZQAHRC
|
6.2 | IC50 | 4 | — | |
TUVMHEGGYLIJHD
|
6.2 | IC50 | 3 | — | |
WCILOMUUNVPIKQ
|
6.2 | IC50 | 5 | — | |
XIMIJJARGYSDBU
|
6.2 | IC50 | 4 | — | |
FRYSEKUUHUUJPX
|
6.2 | IC50 | 3 | — | |
KYFZKWSQWIPREE
|
6.1 | IC50 | 2 | — |