Target Details
| UniProt AC | P41229 |
|---|---|
| Gene Symbol | KDM5C |
| Protein Name | Lysine-specific demethylase 5C |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF01388 (ARID) PF02373 (JmjC) PF02375 (JmjN) PF21323 (KDM5_C-hel) PF00628 (PHD) PF08429 (PLU-1) PF02928 (zf-C5HC2) |
Summary
- Multi-target molecules 108
- Clinical molecules 0
- Avg pChEMBL 6.96
Associated Diseases (1)
Active Molecules (108)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
HJWSLDFYCQJXLZ
|
8.2 | IC50 | 3 | — | |
MZLRXFKOAWCNNY
|
8.2 | IC50 | 3 | — | |
FAOZNCYQMCTIBT
|
7.9 | IC50 | 6 | — | |
ZVDVVBQKFXBYJN
|
7.9 | IC50 | 4 | — | |
DHXKRMSKXLDZGY
|
7.8 | IC50 | 3 | — | |
VQBICUVJQVNKBH
|
7.8 | IC50 | 4 | — | |
AIEULFAFWDPGEJ
|
7.7 | IC50 | 4 | — | |
UZFOOEZHJLPYBL
|
7.7 | IC50 | 4 | — | |
RZAREOJWVVYJGA
|
7.7 | IC50 | 4 | — | |
DDRYBCASNXOENV
|
7.6 | IC50 | 4 | — | |
MIHKHZZRKYZHJU
|
7.6 | IC50 | 4 | — | |
RNTSNXOXDNEYJK
|
7.6 | IC50 | 4 | — | |
BJPPOTJAQZGVIA
|
7.6 | IC50 | 4 | — | |
LNMSTPSCCSYARO
|
7.6 | IC50 | 2 | — | |
BSWSHYUVWCPTHU
|
7.5 | IC50 | 4 | — | |
WAXTXDDUSDCZNA
|
7.5 | IC50 | 4 | — | |
VEDMWPYTXDSWTP
|
7.5 | IC50 | 4 | — | |
XAXOYJMMDIYHQF
|
7.5 | IC50 | 4 | — | |
MQVSMJMODJEBMM
|
7.5 | IC50 | 4 | — | |
LAGKZFNQXIBSDJ
|
7.4 | IC50 | 4 | — | |
FBNVHXXPQQVJCQ
|
7.4 | IC50 | 4 | — | |
LHYVGHNYNLLNOV
|
7.4 | IC50 | 4 | — | |
XIVQRYFYMNIDET
|
7.3 | IC50 | 4 | — | |
YSKANQRCYYKDSC
|
7.3 | IC50 | 4 | — | |
JOPSCFKAECJOQR
|
7.3 | IC50 | 4 | — | |
KWVQXVRPRJIRSJ
|
7.3 | IC50 | 4 | — | |
RLRGPZGIQMEBLC
|
7.3 | IC50 | 4 | — | |
DUTYNXONGTVYED
|
7.3 | IC50 | 4 | — | |
NLYFSJWBMSCWSU
|
7.3 | IC50 | 4 | — | |
CYMWJZQYPTVZRX
|
7.3 | IC50 | 4 | — | |
XWSGXVMUELGWLQ
|
7.3 | IC50 | 4 | — | |
CXEXTVGTDZRKJS
|
7.3 | IC50 | 3 | — | |
FWXNBMPVCHFMRX
|
7.2 | IC50 | 4 | — | |
OKSIGHDJUXBCLG
|
7.2 | IC50 | 4 | — | |
RGGMVQDDHDCRDM
|
7.2 | IC50 | 9 | — | |
IBSVWTKUXPGZFI
|
7.2 | IC50 | 3 | — | |
RIVJXVMWOIAAEH
|
7.2 | IC50 | 4 | — | |
ZTYRLXUTLYBVHH
|
7.2 | IC50 | 8 | — | |
INPKYGJHWGXUDF
|
7.2 | IC50 | 4 | — | |
LDSDVQOOEYCWQS
|
7.2 | IC50 | 4 | — | |
KRXWJZIHQRIGSJ
|
7.2 | IC50 | 3 | — | |
SQDIBEJSOSAPGF
|
7.2 | IC50 | 4 | — | |
PNFMVADNCOGWME
|
7.2 | IC50 | 4 | — | |
ZBLHURFMYIWFIY
|
7.2 | IC50 | 4 | — | |
UAKCGLKAUUAKCL
|
7.1 | IC50 | 4 | — | |
NLGUSOLKPNWPKR
|
7.1 | IC50 | 4 | — | |
AYSIHEFQSAIYGY
|
7.1 | IC50 | 4 | — | |
IALMMJCSQDGXBB
|
7.1 | IC50 | 5 | — | |
TWKOGDIJEBKSKF
|
7.1 | IC50 | 4 | — | |
CLDDHWNJFOWJLH
|
7.1 | IC50 | 4 | — |