Target Details
| UniProt AC | P41180 |
|---|---|
| Gene Symbol | CASR |
| Protein Name | Extracellular calcium-sensing receptor |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00003 (7tm_3) PF01094 (ANF_receptor) PF07562 (NCD3G) |
Summary
- Multi-target molecules 12
- Clinical molecules 0
- Avg pChEMBL 8.11
KEGG Pathways (2)
Associated Diseases (7)
Active Molecules (12)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
WJNQZXPCJCLCNG
|
10.7 | IC50 | 6 | — | |
HOWBDMROKCOABA
|
10.5 | IC50 | 7 | — | |
BKMZXLKUUMOTKA
|
10.2 | IC50 | 3 | — | |
PPLVDBKGJPKXLH
|
8.3 | IC50 | 4 | — | |
PBDMWGSHTOZGOM
|
8.0 | IC50 | 6 | — | |
PYNFKKBWKOSQPJ
|
7.6 | IC50 | 2 | — | |
PZUJQWHTIRWCID
|
7.6 | IC50 | 7 | — | |
DWAKJSOEJNKPME
|
7.2 | IC50 | 2 | — | |
MVYOBBWPCHPRSG
|
7.2 | IC50 | 5 | — | |
KCCUCFUQSYGPBH
|
6.8 | IC50 | 6 | — | |
DWAKJSOEJNKPME
|
6.7 | IC50 | 2 | — | |
DWAKJSOEJNKPME
|
6.5 | IC50 | 2 | — |