Target Details
| UniProt AC | P40337 |
|---|---|
| Gene Symbol | VHL |
| Protein Name | von Hippel-Lindau disease tumor suppressor |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF01847 (VHL) PF17211 (VHL_C) |
Summary
- Multi-target molecules 158
- Clinical molecules 0
- Avg pChEMBL 6.8
KEGG Pathways (4)
Associated Diseases (4)
Active Molecules (158)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
GAUPKVQHAPDXDP
|
6.4 | IC50 | 2 | — | |
PCDKDIQCUMWKIP
|
6.4 | IC50 | 2 | — | |
ZXSIYBHMUJKMEO
|
6.4 | IC50 | 3 | — | |
LZOHYKPBMBVPRQ
|
6.4 | IC50 | 2 | — | |
FKLIIDWOMMJUOM
|
6.4 | IC50 | 2 | — | |
ORYIAYLKBQJOHH
|
6.3 | IC50 | 2 | — | |
YHCWTMCHWMELSK
|
6.3 | Kd | 3 | — | |
CLXVPFKDBLSVPK
|
6.3 | Kd | 3 | — | |
FYSWLIFIYIVHPI
|
6.3 | Ki | 4 | — | |
INXGMIWEZJNJOA
|
6.3 | IC50 | 3 | — | |
LZQIXKMTFOXRIS
|
6.3 | IC50 | 2 | — | |
AQIQXAQNDASVRZ
|
6.3 | IC50 | 6 | — | |
GXUKQNHVGSQLDF
|
6.3 | IC50 | 3 | — | |
JBVJZYKQXUYGRI
|
6.3 | Kd | 3 | — | |
RIEGJNXDHULIKM
|
6.3 | IC50 | 3 | — | |
WHHJTGONFDCQEJ
|
6.3 | Kd | 3 | — | |
LRZZTYVIZNQTND
|
6.3 | IC50 | 2 | — | |
ZPRVCDPVYCHLDT
|
6.3 | Kd | 3 | — | |
AIFXAXRMMBWMAG
|
6.3 | Kd | 4 | — | |
GHPGTOYKAZPYSV
|
6.3 | Kd | 3 | — | |
AILRADAXUVEEIR
|
6.3 | IC50 | 75 | — | |
KFWCDEUBKRIYPP
|
6.3 | IC50 | 2 | — | |
BADMTEFLTGIPRJ
|
6.2 | IC50 | 2 | — | |
RKYJQMJUEDVPPS
|
6.2 | Kd | 3 | — | |
DYUJLNPTOOBZBB
|
6.2 | IC50 | 3 | — | |
STUOLYLKGJYHJO
|
6.2 | IC50 | 2 | — | |
HWJIMIISFDRVKH
|
6.2 | IC50 | 2 | — | |
DZMNNNDNOJMJII
|
6.2 | IC50 | 2 | — | |
GVGRVMHQPPDFKJ
|
6.2 | IC50 | 2 | — | |
PECICTZKVKHDTH
|
6.2 | Kd | 3 | — | |
QEVBIPGACHQDQE
|
6.2 | IC50 | 2 | — | |
HEDFFPYRFJKXQP
|
6.2 | IC50 | 2 | — | |
JKHAXURJIZDRKK
|
6.2 | Kd | 3 | — | |
SEXYQPBYWZVVSL
|
6.2 | IC50 | 2 | — | |
DJTBXBQGAPPXCU
|
6.1 | IC50 | 2 | — | |
YMRFUSDFDQZOFK
|
6.1 | IC50 | 2 | — | |
QZNQKYSTRCIAKT
|
6.1 | Kd | 3 | — | |
BBLUCKCGFGRHBM
|
6.1 | IC50 | 5 | — | |
JYRWFOMSBQFKQQ
|
6.1 | IC50 | 2 | — | |
SDAVNUYOWAVNNJ
|
6.1 | IC50 | 3 | — | |
GENALQNUPMUAKG
|
6.1 | IC50 | 2 | — | |
ILKLJSWMSIMESB
|
6.1 | IC50 | 2 | — | |
NRFUNIWQTXTAPE
|
6.1 | IC50 | 2 | — | |
AQPXPSSVMZCLHW
|
6.1 | IC50 | 2 | — | |
FEEFVTMBJHCHIE
|
6.1 | IC50 | 2 | — | |
GTVIVAIUGKIIDT
|
6.1 | IC50 | 2 | — | |
IHPWGIHQQYLHCE
|
6.1 | IC50 | 2 | — | |
PLSIZPKPMOPGBN
|
6.1 | IC50 | 2 | — | |
PMGOJGGCHPNUEJ
|
6.1 | IC50 | 2 | — | |
WHYNNQMYHZONCV
|
6.1 | Kd | 3 | — |