Target Details
| UniProt AC | P40313 |
|---|---|
| Gene Symbol | CTRL |
| Protein Name | Chymotrypsin-like protease CTRL-1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00089 (Trypsin) |
Summary
- Multi-target molecules 22
- Clinical molecules 0
- Avg pChEMBL 7.43
KEGG Pathways (2)
Active Molecules (22)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
RERFKFYMYKTFND
|
9.4 | Ki | 5 | — | |
RSKAMAUHJHZMQX
|
9.1 | Ki | 6 | — | |
ZBVDAILDYSBUAI
|
8.8 | Ki | 6 | — | |
OOEXUWDNTCTJMI
|
8.7 | IC50 | 20 | — | |
WCAAICVTUFKIIQ
|
8.4 | IC50 | 2 | — | |
IRAOTOKFIWRLCT
|
8.4 | IC50 | 2 | — | |
NMKCXXGHQVJDPK
|
8.2 | IC50 | 20 | — | |
XADHZGACMQLWMK
|
8.0 | Ki | 6 | — | |
URCIFSDWSKDSMC
|
7.7 | IC50 | 2 | — | |
AXXYATYQRMPQSN
|
7.7 | Ki | 6 | — | |
FSWFYCYPTDLKON
|
7.5 | Ki | 9 | — | |
SENRSUXIIOUWCL
|
7.2 | IC50 | 3 | — | |
HQIKQQKBLGAORR
|
6.8 | Ki | 6 | — | |
SWZXEVABPLUDIO
|
6.8 | IC50 | 20 | — | |
FAFKHKDMLVSDPG
|
6.6 | IC50 | 2 | — | |
KKRGXDSPEUYYKM
|
6.5 | Ki | 6 | — | |
XNGYIZWSDCYUOZ
|
6.5 | IC50 | 2 | — | |
IELDEMOVCFANHT
|
6.4 | IC50 | 5 | — | |
RAGGAKACRGQVDL
|
6.4 | IC50 | 2 | — | |
LRHBPVVPFQMQPP
|
6.3 | Ki | 6 | — | |
CPBDFCXKCBYWQN
|
6.2 | IC50 | 5 | — | |
MBGPBHRYFCMIPN
|
6.0 | Ki | 5 | — |