Target Details
| UniProt AC | P39900 |
|---|---|
| Gene Symbol | MMP12 |
| Protein Name | Macrophage metalloelastase |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00045 (Hemopexin) PF00413 (Peptidase_M10) PF01471 (PG_binding_1) |
Summary
- Multi-target molecules 404
- Clinical molecules 97
- Avg pChEMBL 7.52
Active Molecules (404)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
XTJBTJMEXZEGIF
|
7.6 | IC50 | 6 | — | |
SQQRAMLTIHSAJA
|
7.5 | IC50 | 2 | — | |
PFIFGQWOKBQYID
|
7.5 | IC50 | 9 | Yes | |
QPLQAMVXCDXOBY
|
7.5 | IC50 | 5 | — | |
ZTJUBPXNBSLSGL
|
7.5 | IC50 | 6 | Yes | |
QQDWEVONJRXVDB
|
7.5 | Ki | 6 | Yes | |
CTCTZAXBKWKMKL
|
7.5 | Ki | 3 | — | |
ITWGWXCEGHFMHT
|
7.5 | IC50 | 10 | Yes | |
MYWFFXDRJYVELL
|
7.5 | IC50 | 2 | — | |
TUJKFLFRSWBCFZ
|
7.5 | IC50 | 2 | — | |
ZMGHGYMGQVMACZ
|
7.5 | Ki | 3 | — | |
ZXGREOKNJDVFSX
|
7.5 | IC50 | 2 | — | |
LCWWOMJWYGNKJF
|
7.5 | Ki | 2 | — | |
BGPDKPPPOAJAIA
|
7.4 | IC50 | 2 | — | |
MOQWSIABFGAXAW
|
7.4 | IC50 | 5 | — | |
SAIHVCSOGMUZPK
|
7.4 | Ki | 3 | — | |
WKYYIJNBJSICFM
|
7.4 | IC50 | 5 | — | |
FIKHJLBGJKASJJ
|
7.4 | IC50 | 2 | — | |
KHCZZISCPQRODX
|
7.4 | Ki | 6 | Yes | |
OEAKPCGGFWRJFX
|
7.4 | IC50 | 2 | — | |
SBPHMLJEBLNVAI
|
7.4 | IC50 | 3 | — | |
BBPLRBWLQWBZIO
|
7.4 | IC50 | 5 | — | |
LHURUBKIFBZDNZ
|
7.4 | Ki | 3 | — | |
LJOOWNHZCTUDSG
|
7.4 | IC50 | 3 | — | |
XNGFENZBCYVDRR
|
7.4 | IC50 | 2 | — | |
TUUMURVUDGZZQZ
|
7.4 | IC50 | 6 | Yes | |
HDDGWKVPDOMYLP
|
7.4 | Ki | 4 | Yes | |
CPYISUHNJGFCRY
|
7.4 | Ki | 3 | — | |
NKGBFKCCSGHHPF
|
7.4 | IC50 | 2 | — | |
UIVFNXLDHQCJRY
|
7.4 | IC50 | 4 | — | |
YSRLIHTZJHEXLM
|
7.3 | IC50 | 2 | — | |
ZVRMYEBTTBZSJJ
|
7.3 | IC50 | 2 | — | |
JYGPMNNMAQCQMG
|
7.3 | Ki | 4 | — | |
ODKPYAOVENFRFV
|
7.3 | IC50 | 3 | — | |
SMWVRODLVRVTBW
|
7.3 | IC50 | 2 | — | |
VDNQILFFXZGSAK
|
7.3 | Ki | 2 | — | |
HXOLPPZDNXMRHR
|
7.3 | Ki | 4 | — | |
IIRLMDJELCRLPB
|
7.3 | Ki | 3 | — | |
SBKWBGSLOANRHJ
|
7.3 | IC50 | 3 | — | |
YDZNXFWUNLRONX
|
7.3 | IC50 | 4 | — | |
YNSXKATXVIZKSB
|
7.3 | IC50 | 5 | — | |
ZQBDVTJLOHIYJN
|
7.3 | Ki | 2 | — | |
NZUPMMOEPOVBQE
|
7.3 | Ki | 5 | — | |
LWERXEYDLSNPDO
|
7.3 | IC50 | 2 | — | |
GOLLITFKIKKRMV
|
7.2 | Ki | 2 | — | |
YWAKWFLUKNCYMP
|
7.2 | Ki | 2 | — | |
KOVQMCGGWATESY
|
7.2 | Ki | 7 | — | |
MXXLMDWJDJQNCZ
|
7.2 | Ki | 2 | — | |
OVUDWXYTKUKYAX
|
7.2 | IC50 | 9 | Yes | |
YVCCTHCWKOIESX
|
7.2 | IC50 | 8 | Yes |