Target Details
| UniProt AC | P39900 |
|---|---|
| Gene Symbol | MMP12 |
| Protein Name | Macrophage metalloelastase |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00045 (Hemopexin) PF00413 (Peptidase_M10) PF01471 (PG_binding_1) |
Summary
- Multi-target molecules 404
- Clinical molecules 97
- Avg pChEMBL 7.52
Active Molecules (404)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
SKLOAVPDSDQCQV
|
7.9 | IC50 | 2 | — | |
HJFONKSERLWIGE
|
7.8 | IC50 | 4 | Yes | |
IZRGHLXXFQNRMD
|
7.8 | IC50 | 2 | — | |
KKGJFHSYGOMRAH
|
7.8 | IC50 | 2 | — | |
LUHJAOVICRNTRC
|
7.8 | IC50 | 7 | Yes | |
OZAYVSZVQPANBZ
|
7.8 | IC50 | 2 | — | |
QZHAFOIXACHKEM
|
7.8 | IC50 | 5 | — | |
VCJGVCZITQVJET
|
7.8 | Ki | 4 | — | |
VMTJQZUZINLEKC
|
7.8 | IC50 | 5 | Yes | |
BVKYTKVUMKYONQ
|
7.8 | Ki | 5 | — | |
RBZQWZODGBMNHX
|
7.8 | Ki | 6 | Yes | |
MXFJZXDWWXHXMV
|
7.8 | Ki | 7 | — | |
AQWIHDVVCANJLS
|
7.8 | Ki | 3 | — | |
JMWVTDZGNUFBMO
|
7.8 | Ki | 4 | — | |
CUKATAAPVFYVIL
|
7.8 | IC50 | 9 | — | |
FTQOZDRDOVWSBK
|
7.8 | Ki | 3 | — | |
RJKVRZJNTANTQB
|
7.8 | IC50 | 2 | — | |
GWHSSPUFNDIEEQ
|
7.8 | Ki | 4 | — | |
MMIHYNVQXYWTFM
|
7.8 | Ki | 4 | — | |
CKZHFOKQZRZCPF
|
7.8 | IC50 | 9 | Yes | |
ZWXRGJMHGHMUMB
|
7.8 | Ki | 4 | — | |
DDIJQZRWMIFTHG
|
7.8 | IC50 | 3 | — | |
PHBHELQPDZPJEY
|
7.8 | IC50 | 3 | — | |
VIZCCTVYPJKZBP
|
7.8 | IC50 | 3 | — | |
ZSZOBVLJWIXXND
|
7.8 | IC50 | 5 | Yes | |
FFGHBWJVBSUBKN
|
7.7 | IC50 | 2 | — | |
GIEQMQWMJSYCKB
|
7.7 | Ki | 5 | — | |
YWXFICBFTYVHJU
|
7.7 | Ki | 4 | — | |
JVBFGGAYMSJQBZ
|
7.7 | IC50 | 7 | Yes | |
KGICPKKIUBLFER
|
7.7 | Ki | 4 | — | |
LXQUQEBAZBLBEJ
|
7.7 | IC50 | 5 | Yes | |
XBXVQHBAWKNJDL
|
7.7 | IC50 | 2 | — | |
AYFCYVLVRYQGME
|
7.7 | IC50 | 8 | — | |
AYFCYVLVRYQGME
|
7.7 | IC50 | 9 | Yes | |
MZDHADNFNLQINL
|
7.7 | IC50 | 2 | — | |
PEOWGCZHIMSTFM
|
7.7 | IC50 | 2 | — | |
WLZISXXOYYGJNT
|
7.7 | Ki | 12 | Yes | |
QQGKYSPTORHWNZ
|
7.7 | Ki | 6 | — | |
VLFDPMJDVIHWPI
|
7.7 | Ki | 3 | — | |
ZCXHDGANXIWOBA
|
7.7 | IC50 | 3 | — | |
CWDYQHCEZVYJNX
|
7.6 | Ki | 3 | — | |
RQCBSNJRFVZHOS
|
7.6 | IC50 | 10 | Yes | |
WUJPOLIUEWWSHN
|
7.6 | IC50 | 2 | — | |
YEVVFVQVGXPEQO
|
7.6 | Ki | 5 | — | |
NCROEDXPKVIJMH
|
7.6 | IC50 | 2 | — | |
RGCUFTVHLLFSQN
|
7.6 | IC50 | 2 | — | |
ZIKBROOIDUARGQ
|
7.6 | IC50 | 3 | — | |
UWVBDELWTIGPFO
|
7.6 | Ki | 4 | — | |
KSEPBMMZVPGILK
|
7.6 | IC50 | 2 | — | |
OURSUJYXZLSVCS
|
7.6 | IC50 | 5 | — |