Target Details
| UniProt AC | P39900 |
|---|---|
| Gene Symbol | MMP12 |
| Protein Name | Macrophage metalloelastase |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00045 (Hemopexin) PF00413 (Peptidase_M10) PF01471 (PG_binding_1) |
Summary
- Multi-target molecules 404
- Clinical molecules 97
- Avg pChEMBL 7.52
Active Molecules (404)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
IQUZJJXEDANMJD
|
8.1 | Ki | 4 | — | |
IVGHGMHNUBCTDC
|
8.1 | Ki | 6 | Yes | |
NZFXVEQIRZMPRQ
|
8.1 | IC50 | 2 | — | |
OUNOAPVJMCBRTF
|
8.1 | IC50 | 2 | — | |
CKYKLNXMCJIGPN
|
8.1 | Ki | 6 | — | |
ZGSTVUAZFACDLH
|
8.1 | IC50 | 7 | — | |
BMJUABISSDGKOA
|
8.1 | Ki | 6 | — | |
DUPWUQYVKWCUOG
|
8.1 | Ki | 7 | — | |
FAJZOFHZLDUFEM
|
8.1 | Ki | 6 | Yes | |
FQRZOEBSTPAQBJ
|
8.1 | IC50 | 4 | — | |
IWQSGINKBSWILJ
|
8.1 | IC50 | 10 | — | |
LFUNCOOVDREPBK
|
8.1 | Ki | 6 | — | |
UTSFQPTVPZNJJH
|
8.1 | IC50 | 7 | Yes | |
KOVQMCGGWATESY
|
8.1 | Ki | 7 | — | |
CXPHOOFGGKZGTC
|
8.1 | Ki | 5 | — | |
HXZPYZWICHZKRL
|
8.1 | IC50 | 10 | — | |
MNJDNDDQYDSDCH
|
8.1 | IC50 | 2 | — | |
COWAOBZJUFXZPY
|
8.1 | Ki | 2 | — | |
INOYENJSYPDBEC
|
8.1 | IC50 | 3 | — | |
KOVQMCGGWATESY
|
8.1 | Ki | 6 | — | |
KRVMUJILUZQWCW
|
8.1 | IC50 | 2 | — | |
NPTUUUXCZCQNQS
|
8.1 | IC50 | 4 | — | |
TUUMURVUDGZZQZ
|
8.1 | IC50 | 3 | — | |
YJKZJSXUMXIJNB
|
8.1 | Ki | 3 | — | |
ZUGWYJYJZWGIPG
|
8.1 | IC50 | 2 | — | |
PKQOURGVZCVPOK
|
8.0 | IC50 | 2 | — | |
QTXVPJOTKLUYMQ
|
8.0 | IC50 | 5 | — | |
JRZMGNCXDSZZAF
|
8.0 | Ki | 3 | — | |
JXZUMXBHWMKALL
|
8.0 | Ki | 3 | — | |
LMKSZZKXCRCXFM
|
8.0 | Ki | 3 | — | |
YTHUQFQHXZIQRV
|
8.0 | IC50 | 2 | — | |
PASQOFLVNKNUQM
|
8.0 | IC50 | 2 | — | |
QPLRROCTSCFWJD
|
8.0 | IC50 | 2 | — | |
SAJAWNZBKHGJOW
|
8.0 | Ki | 6 | — | |
BICNEVCTASLTLM
|
8.0 | Ki | 6 | — | |
QCVLVTVGVJUODZ
|
8.0 | Ki | 6 | — | |
SKLOAVPDSDQCQV
|
8.0 | IC50 | 2 | — | |
WGKRRJWRVSDOSN
|
8.0 | IC50 | 2 | — | |
YNIHTMMJQXUNPE
|
8.0 | Ki | 7 | Yes | |
IIUXBHAJTPNCIR
|
8.0 | Ki | 6 | — | |
FBDOWURNGYMLPJ
|
7.9 | Ki | 7 | — | |
AEOWLQGPNGMHBP
|
7.9 | Ki | 8 | — | |
RRTBKPAJZZSWKG
|
7.9 | IC50 | 3 | — | |
SIICAQVADMFEDB
|
7.9 | Ki | 8 | Yes | |
TUUMURVUDGZZQZ
|
7.9 | IC50 | 6 | Yes | |
TYZVGHNHMXVHTN
|
7.9 | Ki | 5 | — | |
SJWYFGLDVUQIEF
|
7.9 | Ki | 4 | — | |
BQDVTMRZPWSYOT
|
7.9 | IC50 | 7 | — | |
SQKUIDNBYAHJQB
|
7.9 | IC50 | 5 | — | |
YPLGVMIJHPJLRA
|
7.9 | IC50 | 6 | Yes |