Target Details
UniProt ACP39898
Gene SymbolPMI
Protein NamePlasmepsin I
OrganismPlasmodium falciparum (isolate HB3)
Entry Name
Organism Category Pathogen
Pfam Domains PF00026 (Asp)
Summary
  • Multi-target molecules 150
  • Clinical molecules 0
  • Avg pChEMBL 7.42
Top Co-occurrence Targets
Active Molecules (150)
InChIKey pChEMBL Type Targets Clinical
SXLRRSVMGDBJCS 6.9 IC50 4
OMKLMGOTDGZEAD 6.9 Ki 3
YFDZMWCWLDFBJN 6.8 Ki 2
NUHCGNMIDRXSBS 6.8 Ki 2
VFYYMZZPLBYLND 6.8 Ki 2
FEKNMSKYBGUXQU 6.8 Ki 2
DOFWARZRCWUXKJ 6.7 Ki 2
NDWHOWIMYBKFHZ 6.7 Ki 2
NZOULCSUVJIIAU 6.7 IC50 3
QGSYHABIFFECIP 6.7 Ki 2
TUYZMTOTGANLMU 6.7 Ki 2
YTQGFSGUHSRGSG 6.7 Ki 2
BAFMARVIPPIEQR 6.6 Ki 2
NPGNLTIRWHMQHI 6.6 IC50 3
CDRIGLPEUQNOSZ 6.6 Ki 2
WGQWSPXLSXKUKP 6.6 Ki 2
KKTYZYHUPKXLPL 6.5 IC50 4
KKTYZYHUPKXLPL 6.5 IC50 4
AITYRGXUVZLLCM 6.5 IC50 2
CFMJBMZVLYGUOI 6.5 IC50 4
YKGWCOPGFKGNGN 6.5 IC50 3
MAFOHSLQJYIBJW 6.5 IC50 3
FAIVGEWDQVKBIM 6.5 IC50 3
QLWRZHKNVAZNJS 6.4 IC50 3
IOLYFAMYPGEJGD 6.4 IC50 3
CSSCEUVVFOFENA 6.4 IC50 3
KNBUMBGSBPCJDJ 6.4 Ki 2
FJXRVRLWZPEISE 6.3 IC50 3
GBIFQWZWWHMHND 6.3 Ki 2
WTRBPPZFGGFRNM 6.3 IC50 2
QSSRCISVYCPJDP 6.3 Ki 2
IBSOPQYKTQLOPF 6.2 IC50 4
IFEVIPCVAOYWRW 6.2 IC50 3
BQCVUFHAOOJMIL 6.2 Ki 2
HYDBTWMDIKDHGH 6.2 Ki 2
JJVQUUYZGJWBPW 6.2 IC50 2
KCQAMDDVQXZDMS 6.2 IC50 3
QOFJYJWXEQOHSX 6.2 Ki 2
ZHLPFTVHHADULF 6.2 IC50 4
ZOZZWZVOMAKBJD 6.1 Ki 2
ZOZZWZVOMAKBJD 6.1 Ki 2
MYJBZTCPVQPNGD 6.1 IC50 4
LRPAEQSZBXPQEO 6.1 Ki 2
ZMZTYRZAAPSDOQ 6.1 IC50 3
BQFXWLYPYJMHKI 6.1 IC50 5
KXZKVZPYBMCFET 6.1 IC50 5
HNRLJKSYVDQMAQ 6.1 Ki 2
FSMNBGWEFVUIAV 6.0 IC50 4
HUPMEFWUWBYIQC 6.0 Ki 2
YZGHWKNHLHTVCA 6.0 IC50 2
2D structure