Target Details
UniProt ACP39086
Gene SymbolGRIK1
Protein NameGlutamate receptor ionotropic, kainate 1
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF01094 (ANF_receptor) PF00060 (Lig_chan) PF10613 (Lig_chan-Glu_bd)
Summary
  • Multi-target molecules 44
  • Clinical molecules 0
  • Avg pChEMBL 7.22
Top Co-occurrence Targets
Active Molecules (44)
InChIKey pChEMBL Type Targets Clinical
YUSZFKPLFIQTGF 9.1 Ki 2
VZFRNCSOCOPNDB 9.0 Ki 3
XTASTURWHDUENT 8.7 IC50 2
KRKRAOXTGDJWNI 8.5 Ki 2
OCVKYJFCWLTEPM 8.4 IC50 3
UWBHJOVXAJRYJM 8.4 Ki 2
NAVAGRCBXRSPTH 8.1 Ki 2
IJPARVQEYUOEFX 8.0 IC50 3
JJSGQCLDNBSOPP 7.9 IC50 3
LRUYIRXPCIHVCY 7.9 Ki 2
KNAYYBRIBNEIAL 7.8 Ki 2
QJFJDPVDKZVXJG 7.8 IC50 3
MCAQZDVWMTUXCQ 7.7 Ki 2
JJSGQCLDNBSOPP 7.6 IC50 3
NHFLJQCBAJUWAE 7.5 Ki 3
PJQRHOIDKSEWFE 7.5 Ki 2
FOOYZANHOGCPSP 7.5 Ki 2
OXQXJYQSWZFDBB 7.3 Ki 2
AYWSXMRAQKWRMH 7.3 Ki 3
MKAFLUPVNVGIOL 7.1 Ki 2
YXLQKZHKWIKJKC 7.1 Ki 5
PLUGGALXTRCKCA 7.0 IC50 3
ONWXFZVXNOZZFR 7.0 Ki 9
ROVACBZWABKJSI 7.0 IC50 3
PIWNUFICDRESOQ 7.0 Ki 9
YXQUINDTMKETDY 7.0 Ki 9
ICLSGXPHOMUHDE 6.9 IC50 3
AXIQDNJOMGBWRL 6.9 IC50 3
JJSGQCLDNBSOPP 6.9 IC50 3
TYAXDMDRDFQFHK 6.8 Ki 2
VLSMHEGGTFMBBZ 6.8 Ki 5
DHOYHGUZQYPTFA 6.6 Ki 2
LUIPVVRVNKNJEK 6.6 Ki 5
RCCMXKJGURLWPB 6.6 Ki 4
LRUYIRXPCIHVCY 6.5 Ki 2
WJHKVWNKYRFLBD 6.5 Ki 2
FGLBAJOPAXFWOT 6.4 Ki 2
KTYABWSAGQKAPP 6.3 Ki 9
KXNAWNLNEPJGOW 6.2 Ki 2
WYJNVGSFRNBGEH 6.2 Ki 9
WHUUTDBJXJRKMK 6.2 Ki 5
WHUUTDBJXJRKMK 6.2 Ki 20
UUDAMDVQRQNNHZ 6.1 Ki 5
HMXDWDSNPRNUKI 6.0 Ki 72
2D structure