Target Details
UniProt ACP37288
Gene SymbolAVPR1A
Protein NameVasopressin V1a receptor
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1) PF08983 (V1R_C)
Summary
  • Multi-target molecules 537
  • Clinical molecules 0
  • Avg pChEMBL 7.48
Top Co-occurrence Targets
Active Molecules (537)
InChIKey pChEMBL Type Targets Clinical
NNEUOWNHFVADBM 6.7 Ki 2
PLGWGTWJRMIVMM 6.7 IC50 2
KSNHHKZYKYNBEI 6.7 Ki 6
NUWNAUVHMPVPKS 6.7 Ki 3
SNHJAZWMZSZXFM 6.7 Ki 2
WRNXUQJJCIZICJ 6.7 Ki 3
YHTMCPVKXBVWSY 6.7 Ki 2
CTJMSFRAJDXHHN 6.7 Ki 2
RRHOINWFAMAGIC 6.7 IC50 3
FMJAMEXUMLPVCZ 6.7 Ki 3
JMZJCWNFJOHULV 6.7 Ki 3
BBABDJYQAOTGDM 6.7 Ki 2
UXLBCGXDZQCSQS 6.7 Ki 3
GWCIQCRNPQYHTQ 6.6 IC50 2
LQUBGKQHGZLFAC 6.6 Ki 2
XEJCDFZDXXUIAO 6.6 Ki 3
PBTHEXRSPYUHQA 6.6 IC50 2
XQDRFXUPGZPPOW 6.6 Ki 3
CCDGXHHJZYGCCT 6.6 Ki 3
IIIHGTMRSVLZBO 6.6 Ki 3
IAGBXLVADMVFOS 6.6 Ki 2
HOGUMWHJVRRZNM 6.6 Ki 3
JMGDUUQAXVYNKR 6.6 Ki 2
DFUJBPWYCJPYLU 6.6 IC50 2
FBFXUJQRBJTYOV 6.6 Ki 3
GUNUEYUXARWQNH 6.6 IC50 2
ITRKTGHAVVSQOD 6.6 Ki 3
XZDZYGSNLJCRQP 6.6 Ki 4
BXOKIJAEZHPQKJ 6.5 Ki 2
DMDIUVQYZJYLSL 6.5 IC50 2
OAIPTJXKMLWSCX 6.5 Ki 3
RCIUOILUJSOGMK 6.5 IC50 2
GYHCTFXIZSNGJT 6.5 Ki 4
FCTSOYFQOMNNFT 6.5 IC50 3
HYIUUWYRJRZECB 6.5 IC50 3
IXGKAUJSTHXTMZ 6.5 IC50 2
JOMBFLIRVGBCOV 6.5 IC50 2
LWMAJNMQKFHSBQ 6.5 Ki 2
MBVIKVSCSKQLMV 6.5 IC50 2
NEPDGKSSDURFFD 6.5 IC50 2
NKCUQMHYXYAFEN 6.5 IC50 2
RGFIPTAWXYXPKA 6.5 IC50 3
UNENLVAAGZZQMF 6.5 IC50 2
VQZYMUWBUBIYHT 6.5 IC50 2
BVJZPAJDRJEDNQ 6.5 IC50 2
STJYHFUMHAUIGO 6.5 Ki 2
FLNMCYWWHVDYIM 6.5 Ki 2
OLUJSZLBWZWGJT 6.5 Ki 2
XKQPFXGJKICVEM 6.5 IC50 2
ZYVQPUIRRQVYOK 6.5 IC50 2
2D structure