Target Details
UniProt ACP37288
Gene SymbolAVPR1A
Protein NameVasopressin V1a receptor
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1) PF08983 (V1R_C)
Summary
  • Multi-target molecules 537
  • Clinical molecules 0
  • Avg pChEMBL 7.48
Top Co-occurrence Targets
Active Molecules (537)
InChIKey pChEMBL Type Targets Clinical
JYFKCAWQGRAERG 7.5 IC50 2
AYFSDKAZINYIAF 7.5 Ki 2
KDTFVUGJPCHHNT 7.5 IC50 2
LNQQGRZERBSVFA 7.5 IC50 2
ODSZHEREXLBQGR 7.5 Ki 2
UVTTVOUSHGWOND 7.5 Ki 3
GUDPRPCHKQSPGM 7.5 IC50 2
XBPMJKHKJZYEBV 7.5 IC50 2
OVWKLYGIFZGQOA 7.4 IC50 2
RMXYSWNIIUMPEL 7.4 Ki 4
RMXYSWNIIUMPEL 7.4 Ki 4
JQIGKWPBAVTXQL 7.4 Ki 4
JQIGKWPBAVTXQL 7.4 Ki 4
LQCRQEJXMNDRFQ 7.4 Ki 2
MGZAEJXRAJXGQL 7.4 IC50 2
UILRVXAQZKZLBN 7.4 Ki 3
HLUSMHIRGMOTIA 7.4 Ki 2
DHYIXRVYYFQZFY 7.4 Ki 2
RUQQITPEFZGHMZ 7.4 IC50 2
WACXYFAARRFXRL 7.4 Ki 2
ZATPFKWGNKFRHK 7.4 IC50 2
SRKXXCTZUIJARI 7.4 Ki 2
YFMAYAHNRGYBRU 7.4 Ki 2
VHZTWJGJQKMGFD 7.4 Ki 2
ZHFPIMSXEZPRLC 7.4 IC50 2
GPBATYISDDVOGP 7.4 Ki 2
KVUXXTSFKCYQJS 7.4 Ki 2
VSCHGUOISATNSX 7.4 IC50 2
VXSFROCWTXUWPF 7.4 Ki 2
WACXYFAARRFXRL 7.4 Ki 2
CEKVKDRXUDAAKU 7.4 Ki 2
CYOLRNSRVHAZDY 7.4 Ki 4
JYKTYQLAXRWNPF 7.4 IC50 2
LQIGPRDZPAZFNW 7.4 Ki 2
VCWFFSIHQLCFHS 7.3 IC50 2
GRJNKBDCMVJZIA 7.3 IC50 2
UJKDXGDSNOCPJP 7.3 IC50 2
VFGUUFALPPOHKD 7.3 Ki 2
IFDJPSALQGUKIU 7.3 Ki 3
ISZNHVLTPIWFCQ 7.3 Ki 2
OHQLZPXJQBKSLE 7.3 Ki 2
VPZGCHVXNDFFEJ 7.3 Ki 2
VPZGCHVXNDFFEJ 7.3 Ki 2
BXOKIJAEZHPQKJ 7.3 Ki 2
QFLOUMLKTQRCOG 7.3 IC50 2
RPCBSKXAEBFLCT 7.3 Ki 2
AOIRKVVLTNNALR 7.3 IC50 3
BWMSBDDWGDIHBZ 7.3 IC50 2
DKPKYJWPTURBIV 7.3 Ki 3
FKKQVDLSFNPSNB 7.3 IC50 2
2D structure