Target Details
| UniProt AC | P37288 |
|---|---|
| Gene Symbol | AVPR1A |
| Protein Name | Vasopressin V1a receptor |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00001 (7tm_1) PF08983 (V1R_C) |
Summary
- Multi-target molecules 537
- Clinical molecules 0
- Avg pChEMBL 7.48
KEGG Pathways (5)
Active Molecules (537)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
MZAVMIIYQKZJCP
|
8.4 | IC50 | 2 | — | |
BZWQFQJYEATIKN
|
8.3 | IC50 | 2 | — | |
VTTUVOLMPNOBRT
|
8.3 | IC50 | 2 | — | |
GIPUQWJSEMKBFV
|
8.3 | Ki | 2 | — | |
AVCHIPMGQBIBGJ
|
8.3 | IC50 | 2 | — | |
LDHCZLHYAVCLIP
|
8.3 | IC50 | 2 | — | |
CBWPDTJPGBXARO
|
8.3 | IC50 | 3 | — | |
KZYINFBORHZVKJ
|
8.3 | IC50 | 2 | — | |
SSJBBNZWJHOPCO
|
8.3 | IC50 | 3 | — | |
ZGMNJHJAVDYJPA
|
8.3 | IC50 | 2 | — | |
AHZBXISCIKZVCM
|
8.3 | IC50 | 2 | — | |
VAWQZJUNSPDCQU
|
8.3 | IC50 | 2 | — | |
YBMKUIPFJVPTQV
|
8.3 | Ki | 2 | — | |
OOKXWTMZQKFFDB
|
8.3 | IC50 | 2 | — | |
DVODPQDNNINMKU
|
8.2 | IC50 | 2 | — | |
VDUORTCBRAITLJ
|
8.2 | IC50 | 2 | — | |
UXYNEKLEPXVKQZ
|
8.2 | IC50 | 2 | — | |
BNENBOYVNATGJM
|
8.2 | IC50 | 2 | — | |
GCZOEWZYLOZOQU
|
8.2 | Ki | 2 | — | |
FAGIURAOFFKPDO
|
8.2 | IC50 | 2 | — | |
MMJYONSQOWKBFO
|
8.2 | IC50 | 2 | — | |
GIPUQWJSEMKBFV
|
8.2 | Ki | 2 | — | |
KXIIKZWYFOMDJV
|
8.2 | IC50 | 2 | — | |
LBPVMLAHLBOLKT
|
8.2 | IC50 | 2 | — | |
LDHCZLHYAVCLIP
|
8.2 | IC50 | 2 | — | |
IQZAGSYSVBWEHC
|
8.2 | IC50 | 2 | — | |
OAILZIXLSBGBEW
|
8.2 | Ki | 2 | — | |
QGLQQPXHJMQTAB
|
8.2 | IC50 | 2 | — | |
IYTPQPZUIVPAJS
|
8.2 | IC50 | 2 | — | |
GKRVFJTYBYOXNV
|
8.2 | Ki | 2 | — | |
PRCLJSSODKTIAE
|
8.2 | IC50 | 2 | — | |
URAASRPXIGTYDE
|
8.2 | IC50 | 2 | — | |
IGBXJMWATREZDP
|
8.1 | Ki | 2 | — | |
VMUXNMAOXUZACT
|
8.1 | IC50 | 2 | — | |
XSTBAVMTSHGRBE
|
8.1 | Ki | 2 | — | |
FNCMTVVTRRLGEA
|
8.1 | IC50 | 2 | — | |
GCPCDABXSOXIND
|
8.1 | IC50 | 2 | — | |
QDNRLEGWYUOYCH
|
8.1 | IC50 | 2 | — | |
LAPHLPQSWLATBB
|
8.1 | Ki | 3 | — | |
OOEHNCVFPNJDTF
|
8.1 | IC50 | 2 | — | |
YPBCJEGVEQHBTM
|
8.1 | IC50 | 2 | — | |
MDCQFDQSPQMOFE
|
8.1 | IC50 | 2 | — | |
SRQPDBNJJWQGBP
|
8.1 | IC50 | 2 | — | |
JUNJJZGYUIARTF
|
8.0 | IC50 | 2 | — | |
JYMGVIRSBQVNDW
|
8.0 | IC50 | 2 | — | |
CRPDZUWQFXLWLT
|
8.0 | IC50 | 2 | — | |
VTTUVOLMPNOBRT
|
8.0 | IC50 | 2 | — | |
VTTUVOLMPNOBRT
|
8.0 | IC50 | 2 | — | |
GBOCTZMLOKKIHJ
|
8.0 | IC50 | 3 | — | |
HLCGWRVWUAIGDE
|
8.0 | IC50 | 2 | — |