Target Details
| UniProt AC | P37288 |
|---|---|
| Gene Symbol | AVPR1A |
| Protein Name | Vasopressin V1a receptor |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00001 (7tm_1) PF08983 (V1R_C) |
Summary
- Multi-target molecules 537
- Clinical molecules 0
- Avg pChEMBL 7.48
KEGG Pathways (5)
Active Molecules (537)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
KHQMNMAJGZDPLL
|
8.8 | IC50 | 2 | — | |
ISUZSWPWZCNHEU
|
8.8 | IC50 | 2 | — | |
VFXPCVBUMMROTO
|
8.8 | IC50 | 2 | — | |
BAJYTSHFKZLMBX
|
8.7 | IC50 | 2 | — | |
LLTRIAGHNROFKP
|
8.7 | IC50 | 2 | — | |
QDPVGLNUJIYJDL
|
8.7 | Ki | 2 | — | |
GVTMMJDLFLCNLI
|
8.7 | IC50 | 2 | — | |
DXLYJBKHQDHMEM
|
8.7 | IC50 | 2 | — | |
RUCNKOMMAZUMRZ
|
8.7 | IC50 | 2 | — | |
NQUCSCZUVAWROC
|
8.7 | IC50 | 2 | — | |
KPDNAZVBCCYSTG
|
8.7 | IC50 | 2 | — | |
JTPJNKPWLHDAAT
|
8.7 | Ki | 2 | — | |
JTPJNKPWLHDAAT
|
8.7 | Ki | 2 | — | |
OAILZIXLSBGBEW
|
8.7 | Ki | 2 | — | |
AZXOTZCWQDJCLY
|
8.7 | IC50 | 3 | — | |
PCWMGEPBSLMVKO
|
8.7 | IC50 | 2 | — | |
MVJHCHSVFFDHAX
|
8.7 | Ki | 2 | — | |
RIBXPGIEMRBUDS
|
8.6 | Ki | 3 | — | |
NYRFRZQRJIRSDI
|
8.6 | Ki | 2 | — | |
RUOURPLXVUWWKS
|
8.6 | IC50 | 2 | — | |
QQOZWRPUOVGJDS
|
8.6 | Ki | 2 | — | |
PHOVIPPURLHZTI
|
8.6 | Ki | 3 | — | |
GIPUQWJSEMKBFV
|
8.6 | Ki | 2 | — | |
UWTHWMLQZNPELF
|
8.6 | IC50 | 2 | — | |
CLIPIZUAVXBONL
|
8.5 | Ki | 4 | — | |
CLIPIZUAVXBONL
|
8.5 | Ki | 4 | — | |
UYACBUOCUXQEQZ
|
8.5 | IC50 | 2 | — | |
DJKJVWJQAVGLHJ
|
8.5 | IC50 | 8 | — | |
FYOZKCPPNGGSSM
|
8.5 | IC50 | 2 | — | |
KRCWRSQNQWOWBX
|
8.5 | IC50 | 2 | — | |
LKUCMBNAHQWPJK
|
8.5 | IC50 | 3 | — | |
MEDYXWWEPBZLAH
|
8.5 | Ki | 2 | — | |
FARYFPAIAGOBBI
|
8.5 | Ki | 2 | — | |
QZHOFLRJRNXJMB
|
8.5 | IC50 | 2 | — | |
AHZBXISCIKZVCM
|
8.5 | IC50 | 2 | — | |
POUFGALOZFJHJJ
|
8.5 | IC50 | 2 | — | |
FLKNEUDCRDQUMS
|
8.5 | IC50 | 2 | — | |
VWXRQYYUEIYXCZ
|
8.5 | Ki | 4 | — | |
ZJBBWLNWMSXEGT
|
8.4 | Ki | 2 | — | |
IYDLWKJZWBLCQJ
|
8.4 | IC50 | 2 | — | |
MRGPBAZYRUEDDT
|
8.4 | Ki | 3 | — | |
CVWDILINRDAORG
|
8.4 | Ki | 2 | — | |
GNBCBCRWRBTDTP
|
8.4 | IC50 | 3 | — | |
KULVNZQLXKQFLX
|
8.4 | IC50 | 2 | — | |
MDXNVTZITNMSGJ
|
8.4 | IC50 | 2 | — | |
XNLOKBBHYUNDHJ
|
8.4 | Ki | 2 | — | |
ZAWNCASKMCRQPF
|
8.4 | IC50 | 2 | — | |
AEOQUILQVQWNLS
|
8.4 | IC50 | 2 | — | |
SMYARTHGIPYMLP
|
8.4 | IC50 | 2 | — | |
TXSNKXYGZGTOSS
|
8.4 | IC50 | 2 | — |