Target Details
| UniProt AC | P37288 |
|---|---|
| Gene Symbol | AVPR1A |
| Protein Name | Vasopressin V1a receptor |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00001 (7tm_1) PF08983 (V1R_C) |
Summary
- Multi-target molecules 537
- Clinical molecules 0
- Avg pChEMBL 7.48
KEGG Pathways (5)
Active Molecules (537)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ZEHNRQNEVWJTIS
|
6.2 | IC50 | 3 | — | |
YLVPPCIRFCDKTO
|
6.2 | Ki | 2 | — | |
NECPFYMUAUYSCZ
|
6.1 | Ki | 2 | — | |
NGYIKLFRMYALTL
|
6.1 | IC50 | 2 | — | |
PLAXNJZZHKHVHY
|
6.1 | Ki | 2 | — | |
SBYOJGQINPGOFZ
|
6.1 | Ki | 2 | — | |
TXMAORKGTXFNFB
|
6.1 | Ki | 2 | — | |
HXKFHHNEFCZKPG
|
6.1 | IC50 | 3 | — | |
RSEFMSOKHZWZHB
|
6.1 | Ki | 2 | — | |
VGSQHYIAUDIJTE
|
6.1 | Ki | 3 | — | |
XHLKHNZUBYHMGL
|
6.1 | Ki | 2 | — | |
YOKBGCTZYPOSQM
|
6.1 | IC50 | 4 | — | |
BWZDFVXMWSTRJX
|
6.1 | IC50 | 2 | — | |
KAHSYFRTIXCAIO
|
6.1 | IC50 | 2 | — | |
KCYOYQGEMXQYGQ
|
6.1 | IC50 | 2 | — | |
VFYZZYUWZNJTRX
|
6.1 | IC50 | 2 | — | |
DDPIHYVFODKELW
|
6.1 | IC50 | 2 | — | |
HHWGWPAREUNUGL
|
6.1 | Ki | 2 | — | |
OEFAJMDMCVQKRS
|
6.1 | IC50 | 2 | — | |
LNKKBPHASIKCOF
|
6.1 | Ki | 2 | — | |
WPUYJTITOZWSHH
|
6.1 | IC50 | 3 | — | |
ZJWAEMNLDJQLSS
|
6.1 | Ki | 2 | — | |
DZLVFBJJFCQVAT
|
6.1 | IC50 | 2 | — | |
INGXCNVWWKKWOO
|
6.1 | Ki | 2 | — | |
KJLIRGDIHDNRBJ
|
6.1 | IC50 | 2 | — | |
NDIURTOKKQLXTG
|
6.1 | IC50 | 2 | — | |
RCKPKSSQWGXFSM
|
6.1 | Ki | 3 | — | |
WRHPPQZOFSXDOM
|
6.0 | Ki | 2 | — | |
WUWFMAPHIGQASK
|
6.0 | Ki | 2 | — | |
GZEKBYKHVMXDNP
|
6.0 | Ki | 2 | — | |
HAZIGHWLODGDFY
|
6.0 | IC50 | 3 | — | |
IAGMQISKNISZPR
|
6.0 | IC50 | 3 | — | |
IGNSUDMIGORDMP
|
6.0 | Ki | 2 | — | |
KQIRJHRSAQSCKU
|
6.0 | IC50 | 3 | — | |
LZSJGBRKLXWGBL
|
6.0 | Ki | 2 | — | |
OXCLWDVDHQWXLM
|
6.0 | IC50 | 3 | — | |
RRGQTZFOQQMAOA
|
6.0 | IC50 | 3 | — |